Target Details
| UniProt AC | P08254 |
|---|---|
| Gene Symbol | MMP3 |
| Protein Name | Stromelysin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,292
- Clinical molecules 1086
- Avg pChEMBL 7.4
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (1,292)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VFGGQXYFBRUJJO
|
8.0 | Ki | 3 | Yes | |
YCKAPRALLQTAKS
|
8.0 | IC50 | 6 | Yes | |
YPULLLFYLVWNFW
|
8.0 | Ki | 3 | Yes | |
YQJZTTJHPABLHV
|
8.0 | Ki | 3 | Yes | |
ZQORGANDVNQVJF
|
8.0 | Ki | 6 | Yes | |
DWFUVVZGNJNHKO
|
7.9 | Ki | 7 | Yes | |
NXWFYCXTAINJMY
|
7.9 | Ki | 6 | Yes | |
DTHLOBYXEMQYBV
|
7.9 | Ki | 3 | Yes | |
GKHRDWHFKKUYAX
|
7.9 | IC50 | 8 | Yes | |
GWZMHEYDUOAMNJ
|
7.9 | IC50 | 6 | Yes | |
HDBHDPIRGZHXCM
|
7.9 | IC50 | 4 | Yes | |
HEPINVNDBLHRTM
|
7.9 | IC50 | 6 | Yes | |
HPIJZAVGIHKGTA
|
7.9 | IC50 | 4 | Yes | |
IVPPTWCRAFCOFJ
|
7.9 | IC50 | 5 | — | |
JHUFDQZOUBDJHZ
|
7.9 | Ki | 4 | Yes | |
MHQJDNZHPIZRRV
|
7.9 | IC50 | 4 | — | |
MWYSQPGMUZLIHV
|
7.9 | Ki | 6 | Yes | |
OQWMKRBWGAJEGE
|
7.9 | IC50 | 4 | Yes | |
PJFWFMNFWQFLRK
|
7.9 | Ki | 4 | Yes | |
PTGMPWHDIULCAR
|
7.9 | IC50 | 6 | Yes | |
RVKPGECPCLBLDB
|
7.9 | IC50 | 10 | Yes | |
SPOYPAQQYPYRKF
|
7.9 | Ki | 3 | Yes | |
UJVIDDIDLMDARE
|
7.9 | IC50 | 4 | Yes | |
VCJOCQOXJUMEBE
|
7.9 | IC50 | 6 | Yes | |
XCJPWKHINIJNBZ
|
7.9 | Ki | 4 | Yes | |
DPQCHTZYBRQXQC
|
7.9 | Ki | 7 | Yes | |
QYCUMAKSYBUWER
|
7.9 | Ki | 6 | — | |
DTQSORRPTAWCFK
|
7.9 | Ki | 3 | Yes | |
FAJSWDUTNDYTOS
|
7.9 | Ki | 3 | Yes | |
GUHYZHHGWPARCR
|
7.9 | IC50 | 6 | Yes | |
JGLOGDIUSBZLOV
|
7.9 | IC50 | 3 | Yes | |
LOAUOKWVGGODSI
|
7.9 | IC50 | 3 | Yes | |
PCAPSCAFNCUGDE
|
7.9 | Ki | 6 | Yes | |
RCJJPUINEATAJF
|
7.9 | Ki | 4 | Yes | |
RZFXBBCSOPZCEJ
|
7.9 | Ki | 3 | Yes | |
SJPBXYWXFIQQJH
|
7.9 | Ki | 5 | Yes | |
SRVJEHMEZKLIMK
|
7.9 | Ki | 4 | Yes | |
VUANPBMJTLCNSC
|
7.9 | IC50 | 6 | Yes | |
VXVNMUQIRGITQV
|
7.9 | IC50 | 5 | Yes | |
WIWASQOQNPNFMY
|
7.9 | IC50 | 5 | Yes | |
WXNWNNKHEJMQOM
|
7.9 | IC50 | 8 | Yes | |
GKLAUAGSCYZMQP
|
7.9 | Ki | 7 | Yes | |
XQSIQJLWCRJICL
|
7.9 | Ki | 5 | Yes | |
AILNNKVMFUWMQL
|
7.8 | Ki | 4 | Yes | |
CBDXJWSRGWXYPR
|
7.8 | IC50 | 5 | Yes | |
CHCOTWNQXXEITG
|
7.8 | IC50 | 5 | Yes | |
CYBDDZKSRZPTQR
|
7.8 | IC50 | 6 | Yes | |
HFAGTNGCAZYYLZ
|
7.8 | Ki | 13 | Yes | |
OHBSIIOTSUMCLG
|
7.8 | Ki | 4 | Yes | |
RRLGEVWMENCJGJ
|
7.8 | Ki | 6 | Yes |