Target Details
| UniProt AC | P08254 |
|---|---|
| Gene Symbol | MMP3 |
| Protein Name | Stromelysin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,292
- Clinical molecules 1086
- Avg pChEMBL 7.4
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (1,292)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WXUQPWYPRTYWIR
|
8.1 | IC50 | 6 | Yes | |
KFUADVZPCULIED
|
8.0 | Ki | 5 | — | |
KFUADVZPCULIED
|
8.0 | Ki | 7 | Yes | |
KYOFVPKPPTUVKK
|
8.0 | IC50 | 8 | Yes | |
YKYLOHCKSMYHPL
|
8.0 | IC50 | 6 | Yes | |
DRINIAFHXKEERM
|
8.0 | IC50 | 5 | Yes | |
FYBKBNVRCAQIIE
|
8.0 | Ki | 3 | Yes | |
JHSGRRNCQDDQBC
|
8.0 | IC50 | 9 | — | |
MFDDFJXXVOMZLW
|
8.0 | Ki | 4 | Yes | |
QKXUIPRJJWLPIY
|
8.0 | IC50 | 7 | Yes | |
YPHZFHQBHSELGO
|
8.0 | IC50 | 7 | Yes | |
IKIPPVJMYSOQOD
|
8.0 | IC50 | 6 | Yes | |
MOODLLAARDEUNJ
|
8.0 | Ki | 6 | Yes | |
BGDARAHTNRWTGV
|
8.0 | IC50 | 6 | Yes | |
CPBPQYOAJUZJNL
|
8.0 | IC50 | 7 | Yes | |
DDRBOOUOUSFWET
|
8.0 | IC50 | 4 | — | |
DGFULAROBOKMBD
|
8.0 | Ki | 5 | Yes | |
FMYMFUHWQBEETO
|
8.0 | IC50 | 5 | Yes | |
INVXSBCIDABVMG
|
8.0 | IC50 | 5 | Yes | |
JRJPXBUCHQFJHU
|
8.0 | IC50 | 6 | Yes | |
LTRQYQYXWUQKJZ
|
8.0 | IC50 | 3 | Yes | |
MAVDNGWEBZTACC
|
8.0 | IC50 | 9 | Yes | |
MAVDNGWEBZTACC
|
8.0 | IC50 | 6 | — | |
NAYVOTYJJPROOM
|
8.0 | IC50 | 3 | Yes | |
NKRKWSFHPLAZOP
|
8.0 | IC50 | 7 | Yes | |
NOCFVGZKPITVEY
|
8.0 | IC50 | 5 | Yes | |
NXKGLSOWQLOKML
|
8.0 | IC50 | 3 | Yes | |
NXRASPQMAAGLPZ
|
8.0 | IC50 | 6 | Yes | |
NZVNFHULUBKMQI
|
8.0 | IC50 | 4 | Yes | |
ROVRDWIOAVCKAV
|
8.0 | IC50 | 3 | Yes | |
RTPXKIITNMOTOD
|
8.0 | Ki | 3 | Yes | |
SBIQGLZKCCTUIC
|
8.0 | IC50 | 4 | Yes | |
UAFRGDNTZQMZFA
|
8.0 | Ki | 5 | Yes | |
VPXAENCQUJDPFF
|
8.0 | IC50 | 4 | — | |
XSWDEIOVOAQSMZ
|
8.0 | IC50 | 7 | Yes | |
YLXVWRCBKXEQFD
|
8.0 | IC50 | 6 | Yes | |
YWAPUIQWVUXRRW
|
8.0 | IC50 | 4 | Yes | |
ZAVWWISQYKVWCT
|
8.0 | IC50 | 6 | Yes | |
ZQKGUWOTJVDTGX
|
8.0 | IC50 | 2 | — | |
ZWHGWUJFPYMQHK
|
8.0 | IC50 | 3 | Yes | |
JFMSSTVXWKCAJH
|
8.0 | Ki | 7 | Yes | |
BOCBQLXXKQDYBE
|
8.0 | Ki | 4 | Yes | |
COEWKMGFIMMVCE
|
8.0 | IC50 | 5 | Yes | |
FIAWLFURFKPROF
|
8.0 | IC50 | 7 | Yes | |
LBNAEOGDUCUPFZ
|
8.0 | IC50 | 4 | — | |
LUCWASGSJPPQEE
|
8.0 | IC50 | 3 | — | |
OTEWYJZEFZRZKI
|
8.0 | IC50 | 8 | Yes | |
PZPOCZWOYXDPDG
|
8.0 | IC50 | 5 | Yes | |
REJAGHRLIZEVSB
|
8.0 | IC50 | 5 | Yes | |
UICDMTYNXJBPNZ
|
8.0 | Ki | 4 | Yes |