Target Details
| UniProt AC | P08254 |
|---|---|
| Gene Symbol | MMP3 |
| Protein Name | Stromelysin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,292
- Clinical molecules 1086
- Avg pChEMBL 7.4
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (1,292)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ROSNVSQTEGHUKU
|
8.2 | IC50 | 12 | Yes | |
VBPVZEMPZISXMF
|
8.2 | IC50 | 5 | Yes | |
WLJUNQUGIMIQDZ
|
8.2 | IC50 | 4 | Yes | |
XCMRAHNFEHFBSX
|
8.2 | Ki | 5 | Yes | |
XQXSQQVRMVVPJW
|
8.2 | IC50 | 8 | Yes | |
YBPDYJXZXAPGSU
|
8.2 | IC50 | 6 | Yes | |
ZRDGYJAMDSHROJ
|
8.2 | IC50 | 7 | Yes | |
AHBFOOOWLVWQFO
|
8.1 | IC50 | 6 | Yes | |
AKNDZTHCJLFZCF
|
8.1 | IC50 | 9 | Yes | |
FXEYKJYOHRTUNG
|
8.1 | IC50 | 6 | Yes | |
IPBVPRHDESNKFG
|
8.1 | Ki | 6 | Yes | |
NXBDTIZSKZYBRI
|
8.1 | IC50 | 3 | Yes | |
OHBYAEPYMITRJA
|
8.1 | Ki | 4 | Yes | |
INSQINPAEQOIQL
|
8.1 | IC50 | 7 | Yes | |
DONMTDNLNMLOIC
|
8.1 | Ki | 13 | Yes | |
IOTJDDOXTYOJJN
|
8.1 | IC50 | 6 | Yes | |
SSQXFNKOLMHXPO
|
8.1 | Ki | 6 | Yes | |
GJOCABIDMCKCEG
|
8.1 | IC50 | 5 | Yes | |
IWJCPVCPLCTWHT
|
8.1 | IC50 | 5 | Yes | |
KJBQTISDZZFFDE
|
8.1 | IC50 | 5 | Yes | |
KJQLQEWCQDLQEA
|
8.1 | IC50 | 5 | Yes | |
MDWFJTBWOFNAQX
|
8.1 | IC50 | 7 | Yes | |
MTAVQVITWBDOLI
|
8.1 | Ki | 5 | Yes | |
OCQHJTWHXNLSJE
|
8.1 | IC50 | 5 | Yes | |
RZDQDYGREGZPAT
|
8.1 | IC50 | 5 | Yes | |
SESDSMKBCYCQSU
|
8.1 | IC50 | 6 | Yes | |
UROHLDAMBMAOKL
|
8.1 | IC50 | 5 | Yes | |
WEXOVDYJKZSHRN
|
8.1 | IC50 | 4 | Yes | |
XKUVMLDMSDMUFF
|
8.1 | IC50 | 3 | — | |
XSMMFHYHIAOGPC
|
8.1 | IC50 | 5 | Yes | |
ZGWIOFHKEXLJPC
|
8.1 | IC50 | 5 | Yes | |
ZWDYAHGBOJEURS
|
8.1 | IC50 | 5 | Yes | |
AIBDPCDNFOFGFS
|
8.1 | Ki | 6 | Yes | |
YQELKCVHKSQHTN
|
8.1 | Ki | 5 | Yes | |
AHLWGTUBPHXANM
|
8.1 | Ki | 5 | Yes | |
FMRZZWFHPADOAW
|
8.1 | Ki | 5 | Yes | |
MTRATHZFTCSGDT
|
8.1 | Ki | 6 | Yes | |
YWZDVYPIFZUSBG
|
8.1 | IC50 | 3 | Yes | |
CFUZFFCLLPGACM
|
8.1 | IC50 | 3 | — | |
DZZFIOQATPLRLB
|
8.1 | Ki | 4 | Yes | |
GCBPAPVOMPJQHK
|
8.1 | Ki | 9 | Yes | |
GHWPTWVNZOSEBR
|
8.1 | IC50 | 2 | — | |
HAIGFFSNUYJTQK
|
8.1 | IC50 | 6 | Yes | |
HKGUEYWZKLSNKN
|
8.1 | Ki | 3 | Yes | |
HXNNABWLGZRTMD
|
8.1 | IC50 | 5 | Yes | |
JDOCJRYXQAWUOO
|
8.1 | IC50 | 7 | Yes | |
JQYSJWITJMOASO
|
8.1 | IC50 | 6 | Yes | |
NGILBKZKRQUURV
|
8.1 | IC50 | 5 | Yes | |
PNKICJSNJYXQOE
|
8.1 | IC50 | 3 | — | |
PTONAIKVYGVBIS
|
8.1 | IC50 | 5 | Yes |