Target Details
| UniProt AC | P08254 |
|---|---|
| Gene Symbol | MMP3 |
| Protein Name | Stromelysin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,292
- Clinical molecules 1086
- Avg pChEMBL 7.4
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (1,292)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DZVQTAQHEPKNSI
|
8.2 | IC50 | 6 | Yes | |
ACXYSVKNGLLDLY
|
8.2 | IC50 | 7 | Yes | |
SJVNLZPBUGMURM
|
8.2 | Ki | 3 | Yes | |
SSVAOOCBANMUMS
|
8.2 | IC50 | 5 | Yes | |
DKPQMSLWGNDZTO
|
8.2 | Ki | 5 | Yes | |
FWRANZUQAGPBMV
|
8.2 | Ki | 5 | Yes | |
JJHRUUKMPWUYIB
|
8.2 | IC50 | 5 | Yes | |
AGRDSOUIPBKOKQ
|
8.2 | IC50 | 4 | Yes | |
AJPFDJXQTUJCCW
|
8.2 | Ki | 4 | Yes | |
AKPXMDCVGKJBIP
|
8.2 | Ki | 4 | Yes | |
BJBBGWSFUXQTAD
|
8.2 | IC50 | 2 | — | |
GYHDAVSEPKRYGB
|
8.2 | IC50 | 3 | Yes | |
JBWUJRFOXXRXHG
|
8.2 | IC50 | 5 | Yes | |
NWVCPUQBLORAAX
|
8.2 | IC50 | 3 | — | |
OPSKOPUCTQQUTB
|
8.2 | IC50 | 4 | Yes | |
TZQQXIZDSZWWPC
|
8.2 | IC50 | 6 | Yes | |
VUEMJXMTPAGVNJ
|
8.2 | IC50 | 2 | — | |
WSGLDBYEABEDRD
|
8.2 | Ki | 4 | Yes | |
YIYXDKFJIKECAM
|
8.2 | IC50 | 5 | Yes | |
YNSHKUPPIHHCNP
|
8.2 | IC50 | 6 | Yes | |
FDWJCEDPTNPQLJ
|
8.2 | Ki | 3 | Yes | |
SSFOEYVZLXDDTG
|
8.2 | IC50 | 7 | Yes | |
BUFVDSAQIYWDGD
|
8.2 | Ki | 5 | Yes | |
DGXRLXMZJHBYOU
|
8.2 | Ki | 5 | Yes | |
GAQJSKIBXSLAJK
|
8.2 | IC50 | 6 | Yes | |
KKVTZTBYJGHGCO
|
8.2 | IC50 | 8 | Yes | |
NLAVZJASCRYXPN
|
8.2 | Ki | 5 | Yes | |
VGTPSCHBTJBJOQ
|
8.2 | Ki | 5 | Yes | |
VHCRBJFCQRNNFG
|
8.2 | IC50 | 8 | Yes | |
HTNLSTWGHBHDPS
|
8.2 | IC50 | 8 | Yes | |
TZNUGSCRBFBAFR
|
8.2 | Ki | 7 | Yes | |
VCUJZXCWHYPIIH
|
8.2 | IC50 | 5 | Yes | |
WYWVSRVZNIIISU
|
8.2 | IC50 | 7 | Yes | |
JGHZXBJPZQXVAB
|
8.2 | IC50 | 6 | Yes | |
LXWSFODDORIHFJ
|
8.2 | IC50 | 6 | Yes | |
YYRRVFYCIQQYHU
|
8.2 | Ki | 6 | Yes | |
APCLVQAXJIHPKK
|
8.2 | IC50 | 5 | — | |
DZWVTHAIOWIVNT
|
8.2 | Ki | 7 | Yes | |
KBZNOZAJAJRTII
|
8.2 | IC50 | 10 | Yes | |
OFJQHDDSKOHCOJ
|
8.2 | IC50 | 3 | Yes | |
RNMJVOBQCWORLK
|
8.2 | IC50 | 7 | Yes | |
ANFAAJVPGXQKBB
|
8.2 | IC50 | 6 | Yes | |
CQRAUIRVDKNRIO
|
8.2 | IC50 | 9 | Yes | |
DABGHULKCXXLEE
|
8.2 | IC50 | 4 | — | |
DQXUWRWXYMJLHB
|
8.2 | IC50 | 5 | Yes | |
FIQXBPSAOMLPLJ
|
8.2 | IC50 | 2 | — | |
GJOCABIDMCKCEG
|
8.2 | IC50 | 6 | Yes | |
HXAROWWJPCDNRW
|
8.2 | IC50 | 6 | Yes | |
MTGNBEKVSCTMSE
|
8.2 | IC50 | 5 | Yes | |
QVNUOLHHXUUNEH
|
8.2 | IC50 | 5 | Yes |