Target Details
| UniProt AC | P08254 |
|---|---|
| Gene Symbol | MMP3 |
| Protein Name | Stromelysin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,292
- Clinical molecules 1086
- Avg pChEMBL 7.4
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (1,292)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
REZSPXZZCJTZIK
|
8.4 | IC50 | 8 | Yes | |
REZSPXZZCJTZIK
|
8.4 | IC50 | 6 | — | |
XOOXBIFEOHDRHE
|
8.4 | IC50 | 6 | Yes | |
IFHBUYGFCSEHIF
|
8.4 | IC50 | 6 | Yes | |
JCCRVIZMNYULMQ
|
8.4 | IC50 | 6 | Yes | |
MRZSOAZZNSUPLS
|
8.4 | IC50 | 3 | — | |
MRZSOAZZNSUPLS
|
8.4 | IC50 | 5 | Yes | |
GTBJTISRJIZWKE
|
8.4 | IC50 | 7 | Yes | |
ITYFHVLIAPNWSK
|
8.4 | IC50 | 3 | Yes | |
PTSHMCCZVCAMNJ
|
8.4 | Ki | 6 | Yes | |
AALOSJKQIIRSAO
|
8.3 | IC50 | 6 | Yes | |
FKFABLSWBDUBOL
|
8.3 | Ki | 2 | — | |
LMJBKCLEHMNEQJ
|
8.3 | Ki | 3 | Yes | |
PONKMSIAUNHYAM
|
8.3 | IC50 | 7 | Yes | |
IBUXWZOBVVWCHD
|
8.3 | Ki | 7 | Yes | |
AFLLOSXTZXYSAK
|
8.3 | IC50 | 3 | Yes | |
AGRDSOUIPBKOKQ
|
8.3 | IC50 | 4 | Yes | |
BKIYUSXBJJEODV
|
8.3 | IC50 | 7 | Yes | |
BNESXKYVXODIPJ
|
8.3 | Ki | 4 | Yes | |
BUOKQWSUTKFXOW
|
8.3 | IC50 | 6 | Yes | |
DYBVZAZWVGRLPI
|
8.3 | IC50 | 2 | — | |
GPLRECXXBJTJRJ
|
8.3 | IC50 | 6 | Yes | |
HIYYLOFJQXHPRU
|
8.3 | IC50 | 5 | Yes | |
HTKNWYDCBWYORK
|
8.3 | IC50 | 3 | Yes | |
ITNSNSYBFZWVPE
|
8.3 | IC50 | 5 | Yes | |
JCVSSJUXUIJGBT
|
8.3 | IC50 | 5 | Yes | |
JMKHBHJIGFWJPF
|
8.3 | IC50 | 5 | — | |
NRCQPJPKKZDRND
|
8.3 | Ki | 6 | Yes | |
PDYICDUZWJCQQF
|
8.3 | IC50 | 4 | — | |
PNOYLKIRWUYKLC
|
8.3 | IC50 | 4 | — | |
PRCRNUDMWULKSO
|
8.3 | IC50 | 7 | Yes | |
RLERLGNKRGQTKW
|
8.3 | Ki | 4 | Yes | |
SFESNYSPTLYJFZ
|
8.3 | IC50 | 6 | Yes | |
UKLIIGXGTPSYBF
|
8.3 | IC50 | 8 | Yes | |
YVUNEHSVUBACDW
|
8.3 | IC50 | 6 | Yes | |
ZQJRBAHLNKPYFN
|
8.3 | Ki | 3 | Yes | |
QQWABDFFKSDQLH
|
8.3 | IC50 | 6 | Yes | |
CDUNTBSHRUTDFM
|
8.3 | Ki | 7 | Yes | |
FITSVZFOIGFQQI
|
8.3 | Ki | 6 | Yes | |
QKYPFBUZQDJQHX
|
8.3 | IC50 | 5 | Yes | |
QYFKTMNLZHLRIH
|
8.3 | IC50 | 7 | Yes | |
RBLCSCFFNCADJO
|
8.3 | Ki | 5 | — | |
RBLCSCFFNCADJO
|
8.3 | Ki | 7 | Yes | |
RBLCSCFFNCADJO
|
8.3 | Ki | 5 | — | |
SRBWJOFRJIEWKS
|
8.3 | IC50 | 7 | Yes | |
GMNFREWQYNXZAF
|
8.3 | Ki | 7 | Yes | |
NQHPVFGLBXTGFR
|
8.3 | IC50 | 7 | Yes | |
SSQXFNKOLMHXPO
|
8.3 | Ki | 6 | Yes | |
CIARJCUCRKNXEE
|
8.3 | Ki | 3 | Yes | |
UBPYMHQGZFVTLG
|
8.3 | Ki | 4 | Yes |