Target Details
| UniProt AC | P08254 |
|---|---|
| Gene Symbol | MMP3 |
| Protein Name | Stromelysin-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00045 (Hemopexin) PF00413 (Peptidase_M10) PF01471 (PG_binding_1) |
Summary
- Multi-target molecules 1,292
- Clinical molecules 1086
- Avg pChEMBL 7.4
KEGG Pathways (7)
Associated Diseases (1)
Active Molecules (1,292)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AMVCYHOEVISGQB
|
8.5 | Ki | 4 | Yes | |
AWPBSKGASHYAHG
|
8.5 | IC50 | 5 | Yes | |
BHBDAWJEKOCFGP
|
8.5 | IC50 | 5 | Yes | |
IIKWXGAHGMGLSQ
|
8.5 | IC50 | 3 | — | |
JAKYATQFPKVBNE
|
8.5 | IC50 | 5 | Yes | |
JBYQQXSCANNDNP
|
8.5 | Ki | 4 | Yes | |
JRIUEEGXFJPYTG
|
8.5 | IC50 | 3 | Yes | |
KWXOWVYUSBDBIB
|
8.5 | Ki | 4 | Yes | |
LIQFLIXIOKMDTJ
|
8.5 | Ki | 7 | Yes | |
LTVIJEFEZVFIST
|
8.5 | IC50 | 14 | Yes | |
MAGDFYDBVAIRMV
|
8.5 | IC50 | 3 | — | |
MZIZOOUSSMSGAV
|
8.5 | IC50 | 5 | Yes | |
QGTWMCXPSZIGIN
|
8.5 | IC50 | 6 | Yes | |
QJRFEWMMQFRQAY
|
8.5 | IC50 | 3 | Yes | |
RYMINZKMUZXTLF
|
8.5 | IC50 | 6 | Yes | |
SKUFTRBSRXIMDB
|
8.5 | IC50 | 3 | Yes | |
SXCBCJFEHSPGNX
|
8.5 | Ki | 4 | Yes | |
WYEWOIOFHXNSNW
|
8.5 | Ki | 5 | Yes | |
ZPNXAVJYHSAOKF
|
8.5 | IC50 | 7 | Yes | |
SUSMVCKSLVPRCL
|
8.5 | IC50 | 7 | Yes | |
SUSMVCKSLVPRCL
|
8.5 | IC50 | 5 | — | |
LPRBYIANGHPFSM
|
8.5 | IC50 | 4 | Yes | |
VGAPHGIXAQRVAL
|
8.5 | IC50 | 7 | Yes | |
XVZWTHXPJUVJAU
|
8.5 | IC50 | 6 | Yes | |
GETQXLAMYOMSJS
|
8.5 | IC50 | 8 | Yes | |
SLHHOJZYTMNFRR
|
8.5 | Ki | 7 | Yes | |
SLHHOJZYTMNFRR
|
8.5 | Ki | 6 | Yes | |
TVNINFNNQVBJHI
|
8.5 | IC50 | 8 | Yes | |
WMYJDFANEQLDGP
|
8.5 | IC50 | 6 | — | |
WSWMIGCNSWBCNT
|
8.5 | Ki | 6 | Yes | |
HLOJKFSLAAGGSY
|
8.5 | Ki | 3 | Yes | |
QPEZTCMCOIDQRV
|
8.5 | IC50 | 5 | Yes | |
ZAXDLNVDZOYNCA
|
8.5 | IC50 | 6 | Yes | |
RCXJWFMVFQBLSC
|
8.5 | IC50 | 8 | Yes | |
RYRSPABEKSPRKC
|
8.5 | IC50 | 7 | Yes | |
WHTRIFCXCJYQKX
|
8.4 | IC50 | 3 | Yes | |
WHTRIFCXCJYQKX
|
8.4 | IC50 | 5 | Yes | |
WOZRCMBDSXXEAJ
|
8.4 | Ki | 6 | Yes | |
FLMHRETZLINTLJ
|
8.4 | IC50 | 3 | Yes | |
BJOZETKUSDMMAN
|
8.4 | IC50 | 6 | Yes | |
DRNABTKZDYWZBW
|
8.4 | IC50 | 3 | Yes | |
IIDUBAKXXSWORH
|
8.4 | IC50 | 5 | Yes | |
JVKDGTTXLCSABF
|
8.4 | IC50 | 2 | — | |
JYHCJUBSWRQINP
|
8.4 | IC50 | 3 | Yes | |
LBZOGBFXCHOCBC
|
8.4 | IC50 | 6 | Yes | |
NQPIHEUUYRAYII
|
8.4 | IC50 | 8 | Yes | |
PJTIDEQBVYCKIC
|
8.4 | IC50 | 2 | — | |
WWRZCSYJKWXOGQ
|
8.4 | Ki | 3 | Yes | |
AAMWPNSLYMJRGM
|
8.4 | Ki | 4 | Yes | |
QPPXLNJKZJGLRN
|
8.4 | IC50 | 6 | Yes |