Target Details
| UniProt AC | P08246 |
|---|---|
| Gene Symbol | ELANE |
| Protein Name | Neutrophil elastase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00089 (Trypsin) |
Summary
- Multi-target molecules 90
- Clinical molecules 0
- Avg pChEMBL 7.15
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (90)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JZSOCPVJALRMLO
|
6.9 | IC50 | 2 | — | |
LDFVFAFYMOXYNX
|
6.9 | IC50 | 2 | — | |
OISXGAIRGJIAOA
|
6.9 | Ki | 2 | — | |
PHZGRASPIRNNKM
|
6.9 | Ki | 2 | — | |
UEEPUAFBVYYSEV
|
6.8 | Ki | 2 | — | |
UUKJIEBFYVGYRF
|
6.8 | IC50 | 2 | — | |
UUKJIEBFYVGYRF
|
6.8 | IC50 | 2 | — | |
FUWNGXILMPFYNH
|
6.7 | IC50 | 3 | — | |
LMBCPECAZNCURR
|
6.7 | Ki | 2 | — | |
CNUQWXKBOTXSTQ
|
6.7 | Ki | 2 | — | |
DXPGMMXRSXDODO
|
6.7 | IC50 | 2 | — | |
FUYOZZGSCQXNCB
|
6.7 | IC50 | 3 | — | |
FUYOZZGSCQXNCB
|
6.7 | IC50 | 3 | — | |
JKRQSPIPAUZESC
|
6.7 | IC50 | 2 | — | |
AZZFGWWOGRBVOV
|
6.6 | IC50 | 4 | — | |
DDUSVFYSJIYYFC
|
6.6 | IC50 | 2 | — | |
PSORSGLVGFXCQD
|
6.6 | IC50 | 2 | — | |
OMVZRWSTCVAYPK
|
6.5 | IC50 | 2 | — | |
BYVUBCIRZIXXCV
|
6.5 | IC50 | 2 | — | |
DJBDLEGQGAMIDA
|
6.5 | IC50 | 2 | — | |
UTEFZPPMNAQVQL
|
6.5 | Ki | 2 | — | |
RJVIUDPSQFFUFS
|
6.5 | IC50 | 2 | — | |
SIORZSNWZVSXNL
|
6.5 | Ki | 3 | — | |
CUYVVUGLFUIZAZ
|
6.5 | IC50 | 3 | — | |
CPJZBAKYBNKFMF
|
6.4 | IC50 | 2 | — | |
OXSUHSQWSLABCN
|
6.4 | IC50 | 2 | — | |
BIOAIESFQROFGZ
|
6.4 | IC50 | 2 | — | |
RBWUMQWKDAKXDV
|
6.4 | IC50 | 2 | — | |
WCGUUGGRBIKTOS
|
6.4 | IC50 | 5 | — | |
SQFZQANUUQNKOW
|
6.3 | IC50 | 2 | — | |
JIZUDYAGIUYWQX
|
6.3 | Ki | 2 | — | |
RMVRFXPWQGESLH
|
6.2 | IC50 | 2 | — | |
BBAWEDCPNXPBQM
|
6.2 | IC50 | 9 | — | |
AKHUMVIUALSLOB
|
6.1 | IC50 | 2 | — | |
ATSZLVKWSVRBLA
|
6.1 | IC50 | 4 | — | |
JAXFJECJQZDFJS
|
6.1 | IC50 | 3 | — | |
WRJITTKUXGEQBF
|
6.1 | IC50 | 3 | — | |
DAVZLVYISUEAQE
|
6.0 | IC50 | 2 | — | |
KVKFNRODEGEMQZ
|
6.0 | IC50 | 2 | — | |
KVVHFOADBLGNMS
|
6.0 | Ki | 2 | — |