Target Details
| UniProt AC | P08235 |
|---|---|
| Gene Symbol | NR3C2 |
| Protein Name | Mineralocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 319
- Clinical molecules 10
- Avg pChEMBL 6.93
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (319)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RRDSVYGZMKNAFC
|
6.0 | IC50 | 2 | — | |
VWTXAIVZMCQYKU
|
6.0 | Ki | 3 | — | |
NIJXJFCGNYEYSG
|
6.0 | IC50 | 2 | — | |
WFIFLFARTXGDFP
|
6.0 | IC50 | 2 | — | |
QKBURCBWLIXXPH
|
6.0 | Ki | 2 | — | |
UKKKPJSCGQJZAT
|
6.0 | IC50 | 2 | — | |
MEWQFKSUHJZGCA
|
6.0 | Ki | 4 | — | |
AHCZZOJYVQVLQG
|
6.0 | IC50 | 3 | — | |
POYMYRFGHYKMSL
|
6.0 | IC50 | 4 | — | |
QQGISFDJEJMKIL
|
6.0 | Ki | 3 | — | |
SSAMEZHVGWGDGH
|
6.0 | IC50 | 3 | — | |
IMGXWRKTVOMDLZ
|
6.0 | IC50 | 3 | — | |
KIXSJEJHLVMNMZ
|
6.0 | IC50 | 2 | — | |
NTYALJAURYTROE
|
6.0 | IC50 | 6 | Yes | |
QFRVNOIAPBNRJM
|
6.0 | Ki | 2 | — | |
QGNJUOXZTPPCOF
|
6.0 | IC50 | 3 | — | |
RSVKCRGCARHPAC
|
6.0 | IC50 | 4 | — | |
USLSTEHVCOVPEK
|
6.0 | IC50 | 3 | — | |
XLVWWNSBFIWDGB
|
6.0 | IC50 | 2 | — |