Target Details
| UniProt AC | P08235 |
|---|---|
| Gene Symbol | NR3C2 |
| Protein Name | Mineralocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 319
- Clinical molecules 10
- Avg pChEMBL 6.93
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (319)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BFWRCRIDNKRGTD
|
6.3 | IC50 | 2 | — | |
QAIBFISDVFSRKN
|
6.3 | IC50 | 2 | — | |
AZKXBAPRQCXHRZ
|
6.3 | Ki | 2 | — | |
ARAFJNZXJVLHDR
|
6.3 | IC50 | 3 | — | |
GAKWAQHHESGFAA
|
6.3 | IC50 | 3 | — | |
MKBMFZOEUDKVGZ
|
6.3 | IC50 | 2 | — | |
RXEIQMFFHIVGLD
|
6.3 | IC50 | 3 | — | |
IYIBSFQMWALFFX
|
6.3 | Ki | 2 | — | |
NYAOFNPTQGNQKM
|
6.3 | IC50 | 2 | — | |
OIXUDXUFFGADIZ
|
6.3 | IC50 | 2 | — | |
VPBRSFFMKTUJNN
|
6.3 | IC50 | 2 | — | |
GCBGSMQYZCPYLB
|
6.2 | IC50 | 2 | — | |
CMHJMUZTXMDMKL
|
6.2 | IC50 | 3 | — | |
DJRNAIGSFHOUFL
|
6.2 | IC50 | 2 | — | |
DOSZIFWFKFJGQL
|
6.2 | IC50 | 3 | — | |
IRZVQRHERMOSEM
|
6.2 | Ki | 2 | — | |
PKGWJFNRGGGBJB
|
6.2 | IC50 | 3 | — | |
QPLQDYDXYCUKKE
|
6.2 | IC50 | 3 | — | |
RFZAHUIHPLZLLA
|
6.2 | Ki | 9 | Yes | |
ABDAGDDZOUDCKI
|
6.2 | IC50 | 2 | — | |
DUKSLEMXBDETTE
|
6.2 | IC50 | 2 | — | |
MTJXQXWQRBOMIO
|
6.2 | IC50 | 2 | — | |
CCMNCWDOPDWHKL
|
6.2 | IC50 | 2 | — | |
DCDROSDZJJENGM
|
6.2 | IC50 | 3 | — | |
PCEQNBCVZPRGRR
|
6.2 | IC50 | 3 | — | |
FMZKGKLLLCYGJW
|
6.2 | Ki | 3 | — | |
MJQKPIOTILTXNU
|
6.2 | Ki | 2 | — | |
NTCBYBDADUSXSB
|
6.2 | IC50 | 9 | Yes | |
VYJSUSIGTRGXQC
|
6.2 | IC50 | 3 | — | |
WVCKFHDLPYAJOU
|
6.2 | IC50 | 5 | — | |
AJAOWKDQDBTLKO
|
6.2 | IC50 | 2 | — | |
JLMKYNGLORSHHP
|
6.2 | IC50 | 2 | — | |
KTOKJEZDHROXCU
|
6.2 | IC50 | 2 | — | |
CFDUSNZVLMAHPE
|
6.1 | IC50 | 3 | — | |
JZFUUMIFIPVITG
|
6.1 | IC50 | 2 | — | |
UPKAUNVEGRFAII
|
6.1 | IC50 | 2 | — | |
WCWNFANFHMNQEP
|
6.1 | IC50 | 7 | Yes | |
XZKRNADKQRQVOR
|
6.1 | IC50 | 2 | — | |
JJSZJRHRVRGDNH
|
6.1 | IC50 | 2 | — | |
YROYMPDJQKBNTG
|
6.1 | IC50 | 3 | — | |
VDCNLLFWCBGVMM
|
6.1 | IC50 | 3 | — | |
YFJZCMOHVUUOJJ
|
6.1 | Ki | 3 | — | |
ULOAOMMDFZMTER
|
6.1 | IC50 | 3 | — | |
ADHVTOAGYGEFSM
|
6.1 | IC50 | 2 | — | |
JIKFLEZNTIZKCI
|
6.1 | Ki | 4 | — | |
KDBXYNSMRDJJFO
|
6.1 | IC50 | 2 | — | |
KSBBSPJEGUHNTP
|
6.1 | IC50 | 3 | — | |
KYUGYVXBKPAWOH
|
6.1 | IC50 | 3 | — | |
YUMWHZCQHQAPAQ
|
6.1 | IC50 | 3 | — | |
RQUXQDVRWLHMBG
|
6.0 | IC50 | 2 | — |