Target Details
| UniProt AC | P08235 |
|---|---|
| Gene Symbol | NR3C2 |
| Protein Name | Mineralocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 319
- Clinical molecules 10
- Avg pChEMBL 6.93
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (319)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MGDHDHQGYPSORD
|
6.5 | IC50 | 3 | — | |
PUCKHCPITYMJIM
|
6.5 | IC50 | 2 | — | |
WDXRGPWQVHZTQJ
|
6.5 | IC50 | 5 | — | |
JQMVFHXSBNJQRP
|
6.5 | IC50 | 2 | — | |
JRZWVYSKNVMDLP
|
6.5 | IC50 | 3 | — | |
KLTYQAJNDLZNSD
|
6.5 | IC50 | 2 | — | |
RHQPXBHOFIZXKG
|
6.5 | IC50 | 2 | — | |
VQFLIHCSQSPSJT
|
6.5 | IC50 | 3 | — | |
AZYGKDQZZHOKOM
|
6.5 | IC50 | 2 | — | |
IFNZOVIDIOXFMG
|
6.5 | IC50 | 2 | — | |
VWCZQZNHWPQZGT
|
6.5 | Ki | 3 | — | |
GWBHDCFCUBNVKR
|
6.5 | IC50 | 2 | — | |
KNEYKCUMUCBZNB
|
6.5 | IC50 | 3 | — | |
LCTFQUGGLDHXTH
|
6.5 | IC50 | 3 | — | |
OTKZWGJLFLAVTD
|
6.5 | IC50 | 2 | — | |
KGVGNTCIQIYLQU
|
6.5 | IC50 | 9 | Yes | |
KCVAVMXQQQXOLI
|
6.4 | IC50 | 6 | Yes | |
MPLPTTLNPDVGGI
|
6.4 | IC50 | 2 | — | |
NVKAWKQGWWIWPM
|
6.4 | IC50 | 5 | — | |
DJRNAIGSFHOUFL
|
6.4 | IC50 | 2 | — | |
FEKIYUBTGQLEBI
|
6.4 | Ki | 3 | — | |
HINCRROTVFUICG
|
6.4 | IC50 | 3 | — | |
VPIGGHQZYNIAQH
|
6.4 | IC50 | 2 | — | |
FXSCCOANJPANKE
|
6.4 | IC50 | 3 | — | |
IMDWWFBCGVBAMW
|
6.4 | IC50 | 2 | — | |
KDMGOYHSUFIUAT
|
6.4 | IC50 | 2 | — | |
NNTHLQVZGURUAX
|
6.4 | IC50 | 3 | — | |
YXGACPVGUQXDFZ
|
6.4 | IC50 | 2 | — | |
HFWXCPFGOCGJDK
|
6.4 | IC50 | 3 | — | |
QBUKAFSEUHGMMX
|
6.4 | Ki | 2 | — | |
QOZZBCZFOZCNQK
|
6.4 | IC50 | 3 | — | |
QTOKABCAHAKYAS
|
6.4 | IC50 | 2 | — | |
CFDUSNZVLMAHPE
|
6.4 | IC50 | 3 | — | |
DORQSUNHACTGLQ
|
6.4 | IC50 | 3 | — | |
LRQSPCAZHXKTHC
|
6.4 | Ki | 3 | — | |
SMYUZCJLGBMSME
|
6.4 | IC50 | 3 | — | |
CZOFJQFQALBETE
|
6.4 | Ki | 4 | — | |
FNAPHRONLYQVOG
|
6.4 | IC50 | 2 | — | |
OTWADYHEAKBKQC
|
6.4 | Ki | 4 | — | |
QTOKABCAHAKYAS
|
6.4 | IC50 | 2 | — | |
UGJGTPGLSLQCPP
|
6.4 | IC50 | 3 | — | |
BCWFWNBNYVPLRF
|
6.4 | IC50 | 3 | — | |
KJUOEYJRZUJJLM
|
6.4 | IC50 | 3 | — | |
OPPYDCXBDREGJT
|
6.4 | IC50 | 4 | — | |
BXRDIKRRETWSCY
|
6.3 | IC50 | 2 | — | |
KJOQLFMPAVEWLJ
|
6.3 | IC50 | 3 | — | |
YRAUBPBLFNFPPH
|
6.3 | IC50 | 2 | — | |
AWPVKERKWQLOEG
|
6.3 | IC50 | 4 | Yes | |
FGWOYLFOCSKTSC
|
6.3 | IC50 | 2 | — | |
ADHVTOAGYGEFSM
|
6.3 | IC50 | 2 | — |