Target Details
| UniProt AC | P08235 |
|---|---|
| Gene Symbol | NR3C2 |
| Protein Name | Mineralocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 319
- Clinical molecules 10
- Avg pChEMBL 6.93
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (319)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RSMAEJMIEPTWJC
|
6.8 | IC50 | 2 | — | |
VGCGSAUUQCQDAY
|
6.8 | IC50 | 3 | — | |
ZCEACWHBZXPKIT
|
6.8 | IC50 | 2 | — | |
WFSBONJXUAXVJH
|
6.8 | IC50 | 3 | — | |
XTULMSXFIHGYFS
|
6.8 | IC50 | 3 | — | |
LBBVZEVHJCWQLW
|
6.8 | IC50 | 2 | — | |
NZDONLCAMPFJHQ
|
6.8 | IC50 | 2 | — | |
OMIMAFBBRNJDDU
|
6.8 | IC50 | 3 | — | |
QHSJNOYFBNQNIZ
|
6.8 | IC50 | 2 | — | |
XVYWAUINFAXEKA
|
6.8 | IC50 | 3 | — | |
HINCRROTVFUICG
|
6.7 | IC50 | 3 | — | |
KGFMFEQQZNKWLP
|
6.7 | IC50 | 3 | — | |
SGPHLLUCLSONGK
|
6.7 | IC50 | 2 | — | |
QQFIDVOPZHXZPF
|
6.7 | IC50 | 3 | — | |
XLIGSXQYXJZZSL
|
6.7 | IC50 | 2 | — | |
JFUAWXPBHXKZGA
|
6.7 | IC50 | 2 | — | |
JKBQDIAWGDKQHW
|
6.7 | IC50 | 2 | — | |
WJEDKJKCQOZDNI
|
6.7 | IC50 | 3 | — | |
DGELEWLFMTZTAW
|
6.7 | IC50 | 2 | — | |
ORHHWJMIJCSUTC
|
6.7 | IC50 | 2 | — | |
UCWWMUPWYRSGBY
|
6.7 | IC50 | 2 | — | |
UZSAWQCKBUFFQD
|
6.7 | IC50 | 2 | — | |
JXRAVTIDZDMHLO
|
6.7 | Ki | 4 | — | |
QSDGRHKNICEVHX
|
6.7 | IC50 | 3 | — | |
LIYOMQNHCSVUSQ
|
6.6 | IC50 | 2 | — | |
QTOKABCAHAKYAS
|
6.6 | IC50 | 3 | — | |
JQDUVTPGLRBCNA
|
6.6 | IC50 | 3 | — | |
USMFOMVHIKQVEN
|
6.6 | IC50 | 3 | — | |
QEMGULFBAZGYKI
|
6.6 | IC50 | 2 | — | |
ABDAGDDZOUDCKI
|
6.6 | IC50 | 2 | — | |
HHJSGMINRSKVLO
|
6.6 | IC50 | 3 | — | |
PVUYPBAPWIWFAJ
|
6.6 | IC50 | 2 | — | |
UUIWYLMDKKQBJQ
|
6.6 | IC50 | 3 | — | |
DCRMRSLJFCGKKG
|
6.6 | IC50 | 2 | — | |
JQDUVTPGLRBCNA
|
6.6 | IC50 | 3 | — | |
WSOYYBRZDOKCSB
|
6.6 | IC50 | 2 | — | |
FDMHMFIRHWCKNN
|
6.5 | IC50 | 2 | — | |
NAKVZBYNDIOTLA
|
6.5 | IC50 | 3 | — | |
XZOCWBJVVFJEFU
|
6.5 | IC50 | 2 | — | |
ATJGOPJRRWGHHL
|
6.5 | Ki | 4 | — | |
LEOCLJZACQHETJ
|
6.5 | Ki | 4 | — | |
VPBRSFFMKTUJNN
|
6.5 | IC50 | 2 | — | |
OTNBHAGJVFDFBS
|
6.5 | Ki | 2 | — | |
ALDWINSGSURGLP
|
6.5 | IC50 | 3 | — | |
DLXBCJBMEVKPIX
|
6.5 | Ki | 9 | Yes | |
IDCRMONFSJJBMN
|
6.5 | IC50 | 3 | — | |
USLUSBGRSPWYFF
|
6.5 | IC50 | 3 | — | |
WGGMBWMYJSVPSG
|
6.5 | IC50 | 3 | — | |
AAJNWJFLYOFHIB
|
6.5 | IC50 | 3 | — | |
HKLWSBIHHHYTLH
|
6.5 | IC50 | 2 | — |