Target Details
| UniProt AC | P08235 |
|---|---|
| Gene Symbol | NR3C2 |
| Protein Name | Mineralocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 319
- Clinical molecules 10
- Avg pChEMBL 6.93
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (319)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RNQOQGINTAOCKX
|
7.2 | IC50 | 3 | — | |
ZBEYROVUYHADKP
|
7.2 | IC50 | 2 | — | |
OHUSXUGFNIRYCY
|
7.2 | IC50 | 2 | — | |
NHIKVVXPLBWTNX
|
7.2 | IC50 | 3 | — | |
PKBIAUYNZMVJCB
|
7.2 | IC50 | 2 | — | |
YIJXPXUAVWVXFR
|
7.1 | IC50 | 2 | — | |
OWWJZAKLVDXCMD
|
7.1 | IC50 | 2 | — | |
RBUVZQPMAIWWCG
|
7.1 | IC50 | 2 | — | |
XYFAXIKXGILQET
|
7.1 | IC50 | 2 | — | |
YBDHLGOMHTXGJP
|
7.1 | IC50 | 2 | — | |
HKUKEMRCCWWBFD
|
7.1 | IC50 | 2 | — | |
YGMWYZPIFDQGCI
|
7.1 | IC50 | 3 | — | |
BTEQZWJLBYEBLQ
|
7.1 | Ki | 4 | — | |
HMYGXGUMESBWOB
|
7.0 | IC50 | 2 | — | |
UDQPQRQPOLSCKG
|
7.0 | IC50 | 2 | — | |
DPBAIUSEAGTHBN
|
7.0 | IC50 | 3 | — | |
HIBGPRWWCKCJIN
|
7.0 | IC50 | 3 | — | |
NNEWMMFHUDIZPO
|
7.0 | IC50 | 3 | — | |
NZKHJRBHEWBIFL
|
7.0 | IC50 | 3 | — | |
DKFBPHVUBSXDJB
|
7.0 | IC50 | 3 | — | |
DUZBBWARHFOMBJ
|
7.0 | IC50 | 3 | — | |
NKLKXXWOFGFVKN
|
7.0 | IC50 | 2 | — | |
LVZOQUMLGOHFGL
|
7.0 | IC50 | 3 | — | |
MHWZNBBELRMCAO
|
7.0 | IC50 | 3 | — | |
CEOIQIXVRWVLBN
|
7.0 | IC50 | 3 | — | |
HZRWBHDMULHBAO
|
7.0 | IC50 | 2 | — | |
SFFRJYDGTHMNDH
|
7.0 | IC50 | 3 | — | |
WWTZCUBJPLJNNS
|
7.0 | IC50 | 2 | — | |
FLUKKJOWQPEDIT
|
6.9 | IC50 | 2 | — | |
JKPOACVGQYPLBU
|
6.9 | IC50 | 3 | — | |
KHLLMEXZTPDMCY
|
6.9 | IC50 | 3 | — | |
NXRVYSZNJVQSEI
|
6.9 | IC50 | 2 | — | |
PVYTWCNJUWKUOG
|
6.9 | IC50 | 3 | — | |
MSXMGTMTOVJLOZ
|
6.9 | IC50 | 3 | — | |
YRHKPVJIZXBRCI
|
6.9 | IC50 | 3 | — | |
BBKNEXLBDUPYET
|
6.9 | IC50 | 2 | — | |
WIMXURNPWBOQET
|
6.9 | Ki | 4 | — | |
GIBZLWRPPUSMTC
|
6.9 | IC50 | 4 | — | |
HSLFOYFJYRSLKF
|
6.9 | IC50 | 3 | — | |
VQMSYLLYQOARPD
|
6.9 | IC50 | 3 | — | |
CVFDJBVNXZCLBL
|
6.8 | IC50 | 2 | — | |
ZZWNDPPQMABJJG
|
6.8 | IC50 | 3 | — | |
PYHAWYQXRVXAHX
|
6.8 | Ki | 4 | — | |
ACYYHAZVNHMRMQ
|
6.8 | Ki | 4 | — | |
WMWTYOKRWGGJOA
|
6.8 | IC50 | 4 | — | |
YBIHCFXAMSLIHT
|
6.8 | IC50 | 2 | — | |
ZREYWBOITVVPOZ
|
6.8 | IC50 | 3 | — | |
IFFNOGXSDVOOPK
|
6.8 | Ki | 2 | — | |
WZKWYTSJJZVJLU
|
6.8 | IC50 | 3 | — | |
OZBSREXZWADXQE
|
6.8 | IC50 | 3 | — |