Target Details
| UniProt AC | P08235 |
|---|---|
| Gene Symbol | NR3C2 |
| Protein Name | Mineralocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 319
- Clinical molecules 10
- Avg pChEMBL 6.93
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (319)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZAINQQRFGATLID
|
7.7 | Ki | 4 | — | |
RKFFHZQKHIMLAH
|
7.7 | IC50 | 2 | — | |
FDWPXNLUFQNWMH
|
7.6 | IC50 | 2 | — | |
UTPNUAIWPWLJEC
|
7.6 | Ki | 4 | — | |
NVMGBEWNMCNKHG
|
7.5 | IC50 | 2 | — | |
WDYCDBMOJVBUFD
|
7.5 | IC50 | 3 | — | |
WUXTURZHMMFRPK
|
7.5 | IC50 | 3 | — | |
VXKBREQCYRAEHY
|
7.5 | IC50 | 3 | — | |
AXOMYVRKJFDZJX
|
7.5 | IC50 | 2 | — | |
IMTXAMMYSYUYSB
|
7.5 | IC50 | 2 | — | |
KXMVPYRKURWIPA
|
7.5 | Ki | 4 | — | |
PLOQCPGEMKIJBX
|
7.5 | IC50 | 2 | — | |
JJTJZAROTNIJSJ
|
7.5 | IC50 | 2 | — | |
PORRNAABVGMIRR
|
7.5 | IC50 | 2 | — | |
UREBDLICKHMUKA
|
7.5 | IC50 | 13 | — | |
LPNILISJTWTRLC
|
7.4 | IC50 | 3 | — | |
OIGNJSKKLXVSLS
|
7.4 | IC50 | 7 | — | |
WDXRGPWQVHZTQJ
|
7.4 | Ki | 5 | — | |
FXOBRTHYLJLPSC
|
7.4 | IC50 | 3 | — | |
NDBQYPUELRHJBZ
|
7.4 | IC50 | 2 | — | |
URYARKSTCIJGME
|
7.4 | Ki | 3 | — | |
WDXRGPWQVHZTQJ
|
7.4 | Ki | 5 | — | |
FXUCYRRIEXLTRF
|
7.4 | IC50 | 2 | — | |
CAVTYMQSFAIXRJ
|
7.4 | Ki | 4 | — | |
DORQSUNHACTGLQ
|
7.3 | IC50 | 3 | — | |
SAVAEFOXNWPFKB
|
7.3 | Ki | 3 | — | |
XFLYEUSUDVNPKL
|
7.3 | IC50 | 2 | — | |
YXPRKGBMFPQBDH
|
7.3 | IC50 | 2 | — | |
QFWHAFOCMOQSHC
|
7.3 | IC50 | 3 | — | |
XTLUPLYDVHOHSW
|
7.3 | Ki | 4 | — | |
CBUBLNUCASPVJQ
|
7.3 | IC50 | 2 | — | |
FGCNFOXYZQLPMW
|
7.3 | IC50 | 3 | — | |
PZBXDKKVRHRWOI
|
7.3 | IC50 | 2 | — | |
QCOBTAGFAUBYAO
|
7.3 | IC50 | 2 | — | |
QWWNXNFWXOZGLJ
|
7.3 | IC50 | 3 | — | |
DSSRNDXICGBGMR
|
7.3 | IC50 | 3 | — | |
WMNQFPRREFLTML
|
7.3 | IC50 | 3 | — | |
JGAKOXMSUKTZLQ
|
7.3 | IC50 | 2 | — | |
VRZVKIJRJRBQJT
|
7.3 | IC50 | 4 | — | |
XPEDSWFHLZUGLG
|
7.2 | IC50 | 2 | — | |
BUUOLGKPFRELSS
|
7.2 | IC50 | 3 | — | |
HKLWSBIHHHYTLH
|
7.2 | IC50 | 3 | — | |
HLAUTXJGHQLNRA
|
7.2 | IC50 | 2 | — | |
QMISUBCKEDZHDT
|
7.2 | IC50 | 3 | — | |
YTFZTDYRARTMPD
|
7.2 | IC50 | 2 | — | |
POUMWPFDKBAVDE
|
7.2 | IC50 | 2 | — | |
YGYIVBNMBYBQGZ
|
7.2 | IC50 | 3 | — | |
CPXLOFOGNURDFC
|
7.2 | IC50 | 3 | — | |
MFVGPPNQHPWGHH
|
7.2 | IC50 | 2 | — | |
MQIWXSYBYIIVPE
|
7.2 | IC50 | 3 | — |