Target Details
| UniProt AC | P08235 |
|---|---|
| Gene Symbol | NR3C2 |
| Protein Name | Mineralocorticoid receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00104 (Hormone_recep) PF00105 (zf-C4) |
Summary
- Multi-target molecules 319
- Clinical molecules 10
- Avg pChEMBL 6.93
KEGG Pathways (1)
Associated Diseases (4)
Active Molecules (319)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LGTLOCBNEXITRB
|
9.5 | Ki | 4 | — | |
CZHIJMGMBQCQDA
|
9.4 | Ki | 3 | — | |
NOUXCOKPRXVTDP
|
9.3 | Ki | 4 | — | |
JYGXADMDTFJGBT
|
9.3 | Kd | 4 | — | |
OMFXVFTZEKFJBZ
|
9.3 | Kd | 4 | — | |
PQSUYGKTWSAVDQ
|
9.3 | IC50 | 2 | — | |
CCCIJQPRIXGQOE
|
9.3 | Ki | 4 | — | |
NREZDYQUMMSPNC
|
9.1 | IC50 | 2 | — | |
RINQMJSFPWHRTD
|
9.1 | IC50 | 2 | — | |
UFZZMZCIWOEUKP
|
9.0 | Ki | 4 | — | |
MRSXXYFEMRTFDC
|
8.9 | IC50 | 2 | — | |
MIAURGNSNSBTNK
|
8.8 | Ki | 4 | — | |
SXIDZLMPGLSSSR
|
8.7 | Ki | 4 | — | |
DEFYZGCPPXOTTL
|
8.7 | IC50 | 2 | — | |
NOUXCOKPRXVTDP
|
8.7 | Ki | 3 | — | |
OFYAWCBWRHXDLF
|
8.6 | IC50 | 2 | — | |
LRBFONSWDTXIPJ
|
8.5 | IC50 | 2 | — | |
METQSPRSQINEEU
|
8.5 | IC50 | 3 | — | |
METQSPRSQINEEU
|
8.5 | IC50 | 3 | — | |
OUCNRPREOGLYEL
|
8.4 | IC50 | 2 | — | |
MPFVEJCVRPLSQN
|
8.4 | IC50 | 2 | — | |
ITUJADZBZLVYSO
|
8.4 | IC50 | 2 | — | |
UPCKDXKXFLMNKF
|
8.4 | IC50 | 2 | — | |
ACDLPCXLODOBHE
|
8.3 | IC50 | 3 | — | |
PHIKAOOZNGLKDI
|
8.2 | Ki | 4 | — | |
MIAURGNSNSBTNK
|
8.2 | IC50 | 4 | — | |
NLPNUYHHRWOSGM
|
8.1 | IC50 | 4 | — | |
MIAURGNSNSBTNK
|
8.1 | Ki | 4 | — | |
VKOYHMBQGJRYAN
|
8.1 | IC50 | 3 | — | |
VNDRTKUEQIBKJY
|
8.1 | IC50 | 3 | — | |
XNULRSOGWPFPBL
|
8.0 | IC50 | 2 | — | |
LIHLXWYJHXJFEM
|
8.0 | IC50 | 3 | — | |
UZNBZDTUBTWOBU
|
8.0 | Ki | 4 | — | |
AXXQTTPUMYEBOV
|
8.0 | IC50 | 4 | — | |
CERMKIOTMWNAGM
|
8.0 | IC50 | 2 | — | |
POJKNBHEJAUGMR
|
8.0 | IC50 | 2 | — | |
LXMSZDCAJNLERA
|
7.9 | IC50 | 6 | Yes | |
AXLNGHICNRTHMP
|
7.9 | IC50 | 2 | — | |
RJKFOVLPORLFTN
|
7.8 | IC50 | 10 | Yes | |
VOVIALXJUBGFJZ
|
7.8 | IC50 | 4 | — | |
CLQBRBFJGFBWMS
|
7.8 | IC50 | 3 | — | |
NFAZOJQFTSWUIF
|
7.8 | IC50 | 2 | — | |
NWSIDHCBAFDSKX
|
7.8 | IC50 | 2 | — | |
ZBHGJXVSUFQFPP
|
7.8 | IC50 | 3 | — | |
QLCLQHCJXWSVTF
|
7.8 | IC50 | 3 | — | |
LQJIEYFFKBLJFV
|
7.8 | IC50 | 3 | — | |
FDFMYVGKENHMGM
|
7.8 | IC50 | 2 | — | |
IJTNKDPWHRABRX
|
7.7 | IC50 | 2 | — | |
KAAJYBMWABCTAG
|
7.7 | Ki | 4 | — | |
VXOKHYHZXBLDSC
|
7.7 | Ki | 4 | — |