Target Details
| UniProt AC | P08183 |
|---|---|
| Gene Symbol | ABCB1 |
| Protein Name | ATP-dependent translocase ABCB1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00664 (ABC_membrane) PF00005 (ABC_tran) |
Summary
- Multi-target molecules 62
- Clinical molecules 6
- Avg pChEMBL 6.88
KEGG Pathways (4)
Associated Diseases (3)
Active Molecules (62)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OEIXJPAIZADICN
|
8.7 | IC50 | 3 | — | |
OEIXJPAIZADICN
|
8.7 | IC50 | 3 | — | |
VNMQONKZFZQPCT
|
8.6 | IC50 | 3 | — | |
XPNBVAOZAHYCST
|
8.5 | IC50 | 3 | — | |
VNMQONKZFZQPCT
|
8.5 | IC50 | 3 | — | |
NECCTVFNAYKBCX
|
8.4 | IC50 | 3 | — | |
XPNBVAOZAHYCST
|
8.3 | IC50 | 3 | — | |
HVXBOLULGPECHP
|
8.1 | IC50 | 17 | — | |
ZPFLSSWYPDZJQP
|
7.9 | IC50 | 2 | — | |
GQRFTXWUCZQCHM
|
7.8 | IC50 | 2 | — | |
QMKGFBTVQQZEJM
|
7.5 | IC50 | 2 | — | |
LGGHDPFKSSRQNS
|
7.5 | IC50 | 2 | — | |
LXPCMMVNRMVBIT
|
7.5 | IC50 | 2 | — | |
SGTNSNPWRIOYBX
|
7.4 | IC50 | 19 | — | |
CNPVASHDPUJKPV
|
7.4 | IC50 | 2 | — | |
QFMYKKOZVFBBGI
|
7.4 | IC50 | 2 | — | |
HPVPHZAVNPALGM
|
7.3 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
7.2 | IC50 | 147 | Yes | |
NOOJSKFTZMLHMC
|
7.1 | IC50 | 2 | — | |
HUILBFJFGUWXGF
|
7.1 | IC50 | 2 | — | |
CHAZSVOPUAINSR
|
7.0 | IC50 | 2 | — | |
KQTJIUOOFLJRAY
|
7.0 | IC50 | 2 | — | |
AZSNMRSAGSSBNP
|
7.0 | IC50 | 2 | — | |
JXLYSJRDGCGARV
|
7.0 | Ki | 17 | — | |
NKANXQFJJICGDU
|
7.0 | Ki | 35 | Yes | |
LWMRNOHPZGMUEC
|
7.0 | IC50 | 2 | — | |
IPXHDKAGTKPTNS
|
6.7 | IC50 | 2 | — | |
NRWKOPKPCJMFGI
|
6.7 | IC50 | 2 | — | |
OSFCMRGOZNQUSW
|
6.7 | IC50 | 2 | — | |
LNEPOXFFQSENCJ
|
6.7 | Ki | 33 | Yes | |
RQZREBGUWYXWLE
|
6.7 | IC50 | 2 | — | |
FCDNRJDHYPWDHC
|
6.5 | IC50 | 2 | — | |
GXDALQBWZGODGZ
|
6.5 | IC50 | 21 | Yes | |
SGTNSNPWRIOYBX
|
6.5 | Ki | 2 | — | |
JWHAUXFOSRPERK
|
6.5 | IC50 | 9 | — | |
QKHVBGIOAYREBB
|
6.5 | IC50 | 2 | — | |
WKEBQZAUNGERGA
|
6.5 | IC50 | 2 | — | |
QAGYKUNXZHXKMR
|
6.5 | IC50 | 3 | — | |
QAGYKUNXZHXKMR
|
6.5 | IC50 | 6 | — | |
JCKRZMGEVAGHHV
|
6.5 | IC50 | 2 | — | |
SGTNSNPWRIOYBX
|
6.4 | IC50 | 2 | — | |
LOUPRKONTZGTKE
|
6.4 | Ki | 3 | — | |
VZJNOIQBYQXEEZ
|
6.4 | IC50 | 2 | — | |
WMVUETDQMUIBJX
|
6.3 | IC50 | 2 | — | |
HBGPQWXCRVPJIS
|
6.3 | IC50 | 2 | — | |
DSUWWKJTWPTXFS
|
6.3 | IC50 | 2 | — | |
RJHIEGFHLJUYSA
|
6.3 | IC50 | 5 | — | |
KTUFNOKKBVMGRW
|
6.2 | IC50 | 38 | Yes | |
OLROWHGDTNFZBH
|
6.2 | IC50 | 7 | — | |
ZPEIMTDSQAKGNT
|
6.2 | Ki | 35 | Yes |