Target Details
UniProt ACP08173
Gene SymbolCHRM4
Protein NameMuscarinic acetylcholine receptor M4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 686
  • Clinical molecules 31
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (686)
InChIKey pChEMBL Type Targets Clinical
CNPFYHSXAKKLOF 7.4 Ki 4
RZSWLEFBXTVYMU 7.4 Ki 3
GVTZHKIAVNUTSV 7.4 Ki 4
UNZBDOQVZFAUNP 7.4 Ki 5
PMCCMEISWXQOME 7.3 Kd 5
UXBPYISKBNGZMG 7.3 Ki 4
HNJAEIXPTNJDDI 7.3 Ki 5
SSQJHXZOEJZLAK 7.3 Ki 4
SNSMIIQEKVYNOH 7.3 Ki 5
WJIDIDMJHVMZSA 7.3 IC50 4
IJRUGZIZSARHLR 7.3 Ki 5
LOAZWNRCWBWKAC 7.3 Ki 5
BHAUVKSALKMKRU 7.3 Ki 4
NFVADXLLOOOZIS 7.3 Ki 5
CJGNMVAAMQAWEF 7.3 Ki 16
MVNBPMNELMRFMU 7.3 Ki 5
ORYQYJAEWXGOJB 7.3 Ki 4
CKPSTQITKHNXIA 7.2 Ki 3
MVDUBVLGXGZDSV 7.2 Ki 4
AYQKIBOBFAZBCX 7.2 Ki 5
DIZOCNYCRPRXMN 7.2 Ki 3
XPXPKUQRUOKHFD 7.2 Ki 5
YKICXCKVEJORPH 7.2 Ki 5
KUKJOLRCPDCJAJ 7.2 Ki 5
OMOWOTRKFFNAIT 7.2 IC50 5
PHTUQLWOUWZIMZ 7.2 Ki 7
VMJKUCKTXMESQR 7.2 Ki 5
GLRXSDVYMJTKAU 7.2 Ki 4
IMKYINSUEJXTJZ 7.2 Ki 5
QPNVVIACYJVUOX 7.2 Ki 12
SKEKXGMFLBCYNC 7.2 Ki 5
ITDUNAGUAFBFRA 7.2 Ki 5
LPJZXUYTCJIHTG 7.2 Ki 5
WQILUXNQRKEYJI 7.2 Ki 4
YZCWHHFUBMQIKE 7.2 Ki 5
NASFNLMUWVJIEY 7.2 Ki 5
PBHNZQQGQQOYNM 7.2 IC50 5
RTHXTYWCAPYZGF 7.2 Ki 3
OANBYDFPBWKVGI 7.2 Ki 5
PGDYOGMNQCUWMZ 7.2 IC50 5
XPXPKUQRUOKHFD 7.2 Ki 5
NXIFJNOHOQFSCE 7.1 Ki 5
RAVGDLZWTLVAPH 7.1 Ki 5
ANUNMVJZPWGZDH 7.1 Ki 5
MVWIZZHMSROILD 7.1 Ki 4
GQAHLUHWIIZPFR 7.1 Ki 5
ZPEIMTDSQAKGNT 7.1 Ki 35 Yes
AESSYHBGSGYEPG 7.1 Ki 5
WHZBQLWHOPDIPC 7.1 Ki 5
DMFXETUOWLUQID 7.1 Ki 5
2D structure