Target Details
UniProt ACP08173
Gene SymbolCHRM4
Protein NameMuscarinic acetylcholine receptor M4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 686
  • Clinical molecules 31
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (686)
InChIKey pChEMBL Type Targets Clinical
UQOFGTXDASPNLL 7.6 Ki 3
KXGAHULLQRZYOM 7.6 Ki 5
VPJXQGSRWJZDOB 7.6 Ki 7
AZYYVQIBCPFAIG 7.6 IC50 5
GFDOCHMSKUCLIW 7.6 Ki 5
JOLJIIDDOBNFHW 7.6 Ki 14
KHJKTXKHUACAIJ 7.6 Ki 5
PIVCJDAJTNZQDR 7.6 Ki 3
PUNXWODWMDLZDP 7.6 Ki 5
HJJPJSXJAXAIPN 7.6 Ki 3
KVWDHTXUZHCGIO 7.6 Ki 32 Yes
QTQLWKLZSPZQTO 7.6 Ki 5
OUQAVICYOCWJLG 7.6 Ki 5
AIZMFPJJDXEQKC 7.5 Ki 4
KLBQZWRITKRQQV 7.5 IC50 25 Yes
STUWFURQGSMWES 7.5 Ki 5
UWQNUCNXNKMWKG 7.5 Ki 5
CUYJUFFZSFIMQM 7.5 Ki 5
POGDAPYUQHRUOU 7.5 Ki 5
UFSZYKLBZJNXLV 7.5 Ki 5
XWZQPFIZAGITHQ 7.5 Ki 4
RVTKNIPUELNCNR 7.5 Ki 5
UWVWASPAVBANND 7.5 Ki 5
XCYNAFSXKQRKGO 7.5 Ki 5
LOOAMMHLLVGAEL 7.5 Ki 5
OFBOKKRZVJJZHR 7.5 Ki 5
YSXKPIUOCJLQIE 7.5 Ki 5
AVNRDCQRRUOTCC 7.5 Ki 5
HHXDJDWQQPSWHW 7.5 Ki 4
KRMYNVCNISSHTN 7.5 IC50 2
UNZBDOQVZFAUNP 7.5 Ki 5
YNNUSGIPVFPVBX 7.5 Ki 24 Yes
DIDYGLSKVUKRRP 7.5 Ki 5
GDLIGKIOYRNHDA 7.5 IC50 24 Yes
RMHMFHUVIITRHF 7.5 Ki 5
UFSZYKLBZJNXLV 7.5 Ki 5
RHAFROHARIZTPJ 7.5 Kd 5
MIDPZKJBVKOKKF 7.4 Ki 3
QGJWMGIPVUWDAK 7.4 Ki 5
RPMBYDYUVKEZJA 7.4 Ki 8
XKYMIJTXUGXDLR 7.4 Ki 4
ZTVIKZXZYLEVOL 7.4 IC50 5
DKABYCZEFMBXSO 7.4 Ki 4
DCNMFOFKZLIEDY 7.4 Ki 5
NEUSVAOJNUQRTM 7.4 IC50 13 Yes
OIZGGNJJLMUGKL 7.4 IC50 4
ZFXGEVATMHZGBZ 7.4 Ki 3
JCBGAEQLPPOPDK 7.4 Ki 5
NPDFULBIQZLKSB 7.4 Ki 4
ZYIJZBYORMBFMV 7.4 Ki 3
2D structure