Target Details
UniProt ACP08173
Gene SymbolCHRM4
Protein NameMuscarinic acetylcholine receptor M4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 686
  • Clinical molecules 31
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (686)
InChIKey pChEMBL Type Targets Clinical
SLFGIOIONGJGRT 7.9 Ki 12
GPFBOILGPPNQAT 7.9 Ki 4
KQHKTHFVDIBYJZ 7.9 IC50 5
PKERJUIAPINEEV 7.9 Ki 5
GPFBOILGPPNQAT 7.9 Ki 4
UXBPYISKBNGZMG 7.9 Ki 4
HDAMOICMOAXFLJ 7.9 Ki 4
KLQQZEIBZUZRLW 7.9 Ki 4
MVNBPMNELMRFMU 7.8 Ki 5
OBWGMKKHCLHVIE 7.8 Ki 9
PUYDWHDEVFRQHJ 7.8 Ki 2
VWBQUAMKHIBZSG 7.8 Ki 5
FNCJWKNHUAURLL 7.8 Ki 5
BFELQLHLUNQIHL 7.8 Ki 5
GTJOIOQFIDFYOI 7.8 Ki 4
HATAELBMIJKIHX 7.8 Ki 2
HECAWZFPXYNICY 7.8 Ki 5
IFGIZQGZVWYBFG 7.8 Ki 3
MLPXDKWFNNRLJM 7.8 Ki 4
AVNRDCQRRUOTCC 7.8 Ki 5
GLGYXEJECWKSPZ 7.8 Ki 3
GPFBOILGPPNQAT 7.8 Ki 4
MEAOYGFCVURJIU 7.8 Kd 5
ODQWQRRAPPTVAG 7.8 IC50 20 Yes
VPWKHNIBDCHPNN 7.8 Ki 5
UWKMFEOQWPCWLU 7.8 Ki 5
JNBDSWBJCGQGPV 7.8 Ki 5
BFELQLHLUNQIHL 7.7 Ki 3
GTJOIOQFIDFYOI 7.7 Ki 4
VDDUJINYXKGZLV 7.7 Ki 7
WXPNDRBBWZMPQG 7.7 Ki 28
GPFBOILGPPNQAT 7.7 Ki 4
CLKYBOTWHCENMP 7.7 IC50 5
JDCADUVEQJRIDC 7.7 Ki 5
KFFUMWAFMBSHHP 7.7 Ki 4
SEXKJERBKVAFLC 7.7 Ki 4
SLVMESMUVMCQIY 7.7 Ki 14
ZVNAONQCGLGOAO 7.7 Ki 3
BRMKEVBAZDNRPY 7.7 Kd 5
OGTLDFSTCJABJV 7.7 Ki 5
JETRJUTXVVSGTR 7.7 Ki 4
UUQTXJMGYQWWJC 7.7 Ki 4
VJJVBHULGOMODS 7.7 Ki 3
WKWYANDGYZVVAK 7.7 IC50 4
FPUKGJMTLUQGFZ 7.7 Ki 12
OTYJWRFICHGQJT 7.7 Ki 5
QZUDBNBUXVUHMW 7.7 Ki 39 Yes
HTYJHPPHBQRXGX 7.6 Ki 5
KSKFIMPGQOTLKR 7.6 Ki 5
OHEDKBMQRCAABJ 7.6 IC50 6
2D structure