Target Details
UniProt ACP08173
Gene SymbolCHRM4
Protein NameMuscarinic acetylcholine receptor M4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 686
  • Clinical molecules 31
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (686)
InChIKey pChEMBL Type Targets Clinical
JJCFRYNCJDLXIK 8.2 IC50 25 Yes
WOMCGBFNBSIIEA 8.2 Kd 5
NCPVINAZNPBCKE 8.2 Ki 5
WHKGYJCRLQITBW 8.2 Ki 5
WHKGYJCRLQITBW 8.2 Ki 5
CJRUIOCIHPGNQL 8.2 Ki 5
YUJOQEAGGUIMED 8.2 Ki 5
SQVWTVHVWIHOSU 8.2 Ki 5
BLBSVEUIBHKGSO 8.2 Ki 2
WYDUSKDSKCASEF 8.2 Ki 5
BCUGCHZRMKTPMU 8.1 Ki 6
BEJYISOPDBBZRK 8.1 Ki 4
IXXCPZGOFVCPCH 8.1 Ki 5
KLQQZEIBZUZRLW 8.1 Ki 3
UECHFIXSINCEDW 8.1 Ki 5
AGVQGHLXLYNMSL 8.1 Ki 5
AYFAGRAOJPSHSH 8.1 Ki 19
TYLFZULSDOOCRC 8.1 Ki 5
QTBCATBNRIYMPB 8.1 Ki 5
HXGBXQDTNZMWGS 8.1 Ki 8
KLBQZWRITKRQQV 8.1 Ki 21
RINSDLXTLQIMOU 8.0 Ki 4
XUENORREMLOMPD 8.0 Ki 5
IEEFWRMSEALUNN 8.0 IC50 5
KTWQAWSQSOISLN 8.0 Ki 4
UACRHRRJJCXGPC 8.0 Ki 5
UPPMZCXMQRVMME 8.0 IC50 7
MZDYABXXPZNUCT 8.0 Ki 5
RHKOEKGERJHNJH 8.0 IC50 3
XMDRTFUFPOAGDR 8.0 Ki 9
YLKMPCDZOHNNJU 8.0 IC50 3
KLQQZEIBZUZRLW 8.0 Ki 4
IENFGCJKCCNIMB 8.0 IC50 5
ZMDWHSSHCTZQTD 8.0 Ki 5
BZHQFTZHZVTIMQ 8.0 Ki 5
FMPNFDSPHNUFOS 8.0 Ki 5
FMPNFDSPHNUFOS 8.0 Ki 5
GZXQKCMKEJCSMK 8.0 Kd 5
JYKJJNTVFIWSHT 8.0 Kd 5
PULJCGFLKSMODH 8.0 Ki 5
UPPZIKNLEDOKKO 8.0 Ki 5
UXRUOZRDTXTVAI 8.0 Ki 5
WMIQSPDXASFBFO 8.0 Ki 2
XBBANBCTQDQYBC 8.0 Ki 4
XTLIPTIWGCJFHQ 8.0 Ki 2
ZNXQAFLLESPBNZ 8.0 Ki 5
ZPMRLGPLMNVIDC 8.0 Ki 4
ZUXABONWMNSFBN 8.0 Ki 29
HTYJHPPHBQRXGX 8.0 Ki 5
NGKTYFBTWFLIRS 7.9 Ki 4
2D structure