Target Details
UniProt ACP08173
Gene SymbolCHRM4
Protein NameMuscarinic acetylcholine receptor M4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 686
  • Clinical molecules 31
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (686)
InChIKey pChEMBL Type Targets Clinical
PXHIFOLPKHLYBX 8.6 Ki 5
ROEXPZFFOZZHOY 8.6 Ki 5
XFGSFWFIJFNGQY 8.6 Ki 5
KKEGQSSUXOGEAF 8.6 Ki 5
NEOMSSISKDUIHW 8.6 Ki 3
QRUXDRCXIGZTGT 8.6 Ki 5
XIQVNETUBQGFHX 8.6 Ki 10
FZSXJAWJJQIXFV 8.5 Ki 3
LSMMQGJPNNFZFL 8.5 Ki 3
ZYBBUFPKZJQNLL 8.5 Ki 3
GMLQVLRORNVELR 8.5 Ki 5
OOGJQPCLVADCPB 8.5 Ki 9
QCUQACXEVHRHIF 8.5 Ki 5
DTQIXKQBUYCCQM 8.5 Ki 3
NPNXPJMTHYXCHW 8.5 Ki 4
PMNZXPJWRDBQSA 8.5 Ki 5
NEQYHZCZFMESJN 8.5 Ki 5
OYXCACHCXKHEOC 8.5 Ki 5
UJXAGMVNACHDOG 8.5 Ki 5
XFUPPJKGZWWZGD 8.5 Ki 3
AFLBGAQHDSOPKA 8.5 Ki 5
BGDKAVGWHJFAGW 8.5 Ki 7
DLMOQVWYEFDOHH 8.5 Ki 5
DPWACXBREFHUKJ 8.5 Ki 3
PCEDEEWEONTUHP 8.4 Kd 5
ICZVKTVMHVHOQI 8.4 Ki 5
RTVAKAAPGHVGBW 8.4 Ki 5
GXQAMXKWCFMGON 8.4 Ki 3
ONOZLVJQXQZLPL 8.4 Ki 5
STECJAGHUSJQJN 8.4 IC50 5
STECJAGHUSJQJN 8.4 IC50 4
GKEOHNSBCHXZOA 8.4 Ki 3
MVNBPMNELMRFMU 8.4 Ki 5
OUVBYPZNWMJZAC 8.4 Ki 2
YFWMVRIRFFWDJL 8.4 Ki 5
ITSKPCHXUYILTR 8.4 IC50 3
MNGBIMWSQDCYMU 8.4 Ki 3
AVNRDCQRRUOTCC 8.4 Ki 5
OMZFQPGNVMBMTP 8.4 Ki 3
IJOGXSLRDLSTOS 8.4 Ki 3
HLBJQGCUNYZLFQ 8.3 Ki 4
QBBZFMTXELSEFR 8.3 Ki 2
OANBYDFPBWKVGI 8.3 Ki 5
GIJXKZJWITVLHI 8.3 IC50 4
QZQDZBWQUNVCFF 8.3 Ki 5
GZIIELZICVUEPK 8.3 Ki 5
PCEDEEWEONTUHP 8.3 Kd 5
HWHLPVGTWGOCJO 8.3 Ki 6
ZRYHPQCHHOKSMD 8.3 Ki 4
FZXSXMYFIZKXPT 8.2 Ki 12
2D structure