Target Details
UniProt ACP08173
Gene SymbolCHRM4
Protein NameMuscarinic acetylcholine receptor M4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 686
  • Clinical molecules 31
  • Avg pChEMBL 7.36
Top Co-occurrence Targets
Active Molecules (686)
InChIKey pChEMBL Type Targets Clinical
LERNTVKEWCAPOY 10.8 IC50 5
UKXSKSHDVLQNKG 10.4 Ki 5
GWAMGWDJCYIREE 10.3 Kd 20
IWBMAAUPHUCYCI 10.3 Kd 20
MODBIBJHAWXYOZ 10.3 Kd 20
ZRQMUCDHVVOENY 10.3 Kd 17
NDXFHBBFUCQHAL 10.2 Ki 5
XXWOCVWJOICKHA 10.1 Kd 5
OLZRBZLJTKELRL 10.1 Ki 4
WGOJWDWKHJHXSV 9.9 Ki 5
WOMCGBFNBSIIEA 9.9 Ki 5
LZCOQTDXKCNBEE 9.8 Ki 5
LERNTVKEWCAPOY 9.8 IC50 6
ANGKOCUUWGHLCE 9.8 IC50 5
ASMXXROZKSBQIH 9.7 IC50 5
HGMITUYOCPPQLE 9.7 Ki 5
WOMCGBFNBSIIEA 9.6 Ki 5
OLZRBZLJTKELRL 9.5 Ki 4
OFTJLQGRWRVUFL 9.5 Ki 4
RKUNBYITZUJHSG 9.5 Ki 5
OLYUOAVKDLVFLJ 9.5 Ki 5
OEXHQOGQTVQTAT 9.4 Ki 5
PHRZGNXUUFTVSE 9.4 Ki 5
PHRZGNXUUFTVSE 9.4 Ki 5
XHKPKSGPVFYQNR 9.4 IC50 2
QOJBMAYEUGMTTA 9.3 Ki 5
XXWOCVWJOICKHA 9.3 Kd 5
AFLBGAQHDSOPKA 9.3 Ki 5
DJOCICQNBMTMNG 9.3 Ki 5
OEXHQOGQTVQTAT 9.3 Ki 5
JGOIBENTSQHWDQ 9.2 Ki 5
XHKPKSGPVFYQNR 9.2 IC50 2
HYJRTXSYDAFGJK 9.2 Ki 5
QOXJSXPGWIRRNX 9.2 Ki 5
OTOMMRFOLVUTLQ 9.2 Ki 3
DJOCICQNBMTMNG 9.2 Kd 2
UFSZYKLBZJNXLV 9.2 Ki 5
WCMVSMOIDILBOJ 9.2 Ki 5
VQESBLKWYKQKCC 9.1 Ki 3
PHCOXGCMPCMSJB 9.1 Ki 3
INEDRTXKDAPQKU 9.1 Ki 5
GHHSRBSZNGGGPF 9.1 Ki 3
UOKGNINOAYOIDX 9.1 Ki 5
QJBDLOQOXGQJTD 9.1 Ki 5
BMNOFIWIZFZYES 9.1 Ki 5
WCMVSMOIDILBOJ 9.1 Ki 5
WCMVSMOIDILBOJ 9.1 Ki 5
MMUOGZOUFNQXMP 9.1 Ki 5
RKUNBYITZUJHSG 9.1 Ki 7
PIBNOUQILXRVNG 9.0 Ki 5
2D structure