Target Details
UniProt ACP08172
Gene SymbolCHRM2
Protein NameMuscarinic acetylcholine receptor M2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,645
  • Clinical molecules 27
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,645)
InChIKey pChEMBL Type Targets Clinical
UWKMFEOQWPCWLU 8.0 Ki 5
KQCRPVVAJACIHG 8.0 Ki 3
MVDUBVLGXGZDSV 8.0 Ki 4
BMNOFIWIZFZYES 8.0 Ki 5
UACRHRRJJCXGPC 8.0 Ki 5
FFWZAKHCGSHEHR 8.0 Ki 2
OANBYDFPBWKVGI 8.0 Ki 5
ONOZLVJQXQZLPL 8.0 Ki 5
AFEXNFIIGBMTBH 8.0 Ki 2
FMPNFDSPHNUFOS 8.0 Ki 5
GIJXKZJWITVLHI 8.0 IC50 16
GMGHBSHBCGMTKY 8.0 IC50 3
GNEIWNURFQPOMA 8.0 IC50 3
GPARJKKXMHOXEG 8.0 IC50 2
POIIDLJXIAHDFT 8.0 Ki 5
SADFFAQSWHTWLL 8.0 Ki 5
UXEIWFVTAFVRHB 8.0 Ki 6
YYEWXNWXUYYCSF 8.0 IC50 3
AVNRDCQRRUOTCC 8.0 Ki 5
ZMDWHSSHCTZQTD 8.0 Ki 5
BZHQFTZHZVTIMQ 8.0 Ki 5
FMPNFDSPHNUFOS 8.0 Ki 5
GTJOIOQFIDFYOI 8.0 Ki 4
GZXQKCMKEJCSMK 8.0 Kd 5
INNRKNITHWITSQ 8.0 Ki 3
IPPGGAXXAKWHHQ 8.0 Ki 5
JOMFXRAREZYSMG 8.0 Ki 5
JYKJJNTVFIWSHT 8.0 Kd 5
PNLHOADYGQJVLG 8.0 IC50 3
QCOZXCKWZLHYKC 8.0 Ki 4
UXRUOZRDTXTVAI 8.0 Ki 5
WRRKXJXJKFCUCR 8.0 IC50 3
SPWGJUOMJHFGMM 7.9 Ki 2
XIQVNETUBQGFHX 7.9 Ki 10
AIMDAESTPOXUBL 7.9 Ki 2
DMQAXIJUTYJHIV 7.9 Ki 6
FWARLZJUQIRKFD 7.9 Ki 3
MASSECXUPYPQEW 7.9 Ki 2
NYFXIMCEKNFZKB 7.9 Ki 2
QRCXIALXHOWWTK 7.9 Ki 3
UFSZYKLBZJNXLV 7.9 Ki 5
UQSRLNYPAPLJBP 7.9 IC50 3
XCSJIKDLUXGHQG 7.9 Ki 4
YRSAORSZRHRWKF 7.9 Ki 2
YTSWRFHHGNPXRN 7.9 Ki 3
ZNXQAFLLESPBNZ 7.9 Ki 5
GGJSWQALDWFCMN 7.9 Ki 2
CHCFFXBWNOXOJJ 7.9 IC50 3
GUPWBMMEJNAFFT 7.9 IC50 3
HNJOKNBVVXSFPS 7.9 IC50 2
2D structure