Target Details
UniProt ACP08172
Gene SymbolCHRM2
Protein NameMuscarinic acetylcholine receptor M2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,645
  • Clinical molecules 27
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,645)
InChIKey pChEMBL Type Targets Clinical
NBVYRBDIADJELP 8.6 Ki 2
RTVAKAAPGHVGBW 8.6 Kd 5
YRAPYXYTEMMURR 8.6 Ki 3
BOXHESMXGWQKOM 8.6 IC50 2
CNXWAYYAICBSCA 8.6 IC50 3
DZIWUHCUDURPKK 8.6 IC50 3
GKNPSSNBBWDAGH 8.6 Ki 2
OIVUQKJVYIDTLN 8.6 Ki 2
PIVCJDAJTNZQDR 8.6 Ki 3
DUUCBMCTCKTDOL 8.6 Ki 2
JCZWHTSVKJZFOP 8.6 Ki 2
RTMQZXMBCBMCJK 8.6 Kd 2
DFCLHAWGKPEFIX 8.6 Ki 5
UJXAGMVNACHDOG 8.6 Ki 5
DAIWBMZPSVQRCH 8.6 IC50 3
KKEGQSSUXOGEAF 8.6 Ki 5
AHQFYDVLGIPHDD 8.5 Ki 3
YGBFXINLTZYAPY 8.5 Ki 2
IENFGCJKCCNIMB 8.5 Kd 5
QCUQACXEVHRHIF 8.5 Ki 5
RINSDLXTLQIMOU 8.5 Ki 4
ALYOAWZYSZLYLO 8.5 IC50 2
INEDRTXKDAPQKU 8.5 Ki 5
LYQGZYIUMYUMCO 8.5 IC50 2
XELSLLUJXUXNOB 8.5 Ki 2
VDLFTAVQHMFQHW 8.5 Ki 2
ZGAIDOGAKIQCJU 8.5 IC50 3
NEQYHZCZFMESJN 8.5 Ki 5
PRPBOUUIRMITJF 8.5 Ki 3
STECJAGHUSJQJN 8.5 Ki 4
AFLBGAQHDSOPKA 8.5 Ki 5
CBUABSHDAKLYKZ 8.5 Ki 3
GUWDPEQJYFKDCE 8.5 Ki 3
GPFBOILGPPNQAT 8.5 Ki 4
STECJAGHUSJQJN 8.5 Ki 5
ZVNAONQCGLGOAO 8.5 Ki 3
PCEDEEWEONTUHP 8.4 Kd 5
DCNMFOFKZLIEDY 8.4 Ki 5
GTJOIOQFIDFYOI 8.4 Ki 4
MAGHIFWNWZHPQG 8.4 Ki 5
BDLKVZCRRROJRY 8.4 IC50 3
KBNPGVPUYYZVTB 8.4 Ki 3
BFELQLHLUNQIHL 8.4 Ki 5
HYJRTXSYDAFGJK 8.4 Ki 5
POQGBGCVTONHDT 8.4 Ki 2
RKAJVTVMICVPJE 8.4 IC50 3
BATVXAHTJHXAJQ 8.4 IC50 3
CTFDKSWRIMHOOV 8.4 Kd 3
GPFBOILGPPNQAT 8.4 Ki 4
GRIVDARKNIXUML 8.4 IC50 3
2D structure