Target Details
UniProt ACP08172
Gene SymbolCHRM2
Protein NameMuscarinic acetylcholine receptor M2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,645
  • Clinical molecules 27
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,645)
InChIKey pChEMBL Type Targets Clinical
VBKBVALDNMYEBZ 8.9 Kd 2
QDDPQJCCXUPHKY 8.9 Ki 2
QKMUXXQVPOBBPT 8.9 Ki 3
XVOCHVRQMXWEQB 8.9 Ki 2
WTRLYZUEDFZGKI 8.9 Ki 5
GIXUITONJFXENE 8.8 Ki 2
MNHIAFLMHVAZPM 8.8 Ki 3
SPCFAZXKBQPYBW 8.8 Kd 3
FZOPOAUKSIMGRQ 8.8 Ki 2
RKUNBYITZUJHSG 8.8 Ki 7
WCMVSMOIDILBOJ 8.8 Ki 5
JNBDSWBJCGQGPV 8.8 Ki 5
HDAMOICMOAXFLJ 8.8 Ki 4
FWPIWVUMKDFZSR 8.8 IC50 3
JFEFOFYHVIMFRD 8.8 Kd 3
NYFXIMCEKNFZKB 8.8 Ki 2
OQPFNGUGJOSTMX 8.8 Ki 2
VBKBVALDNMYEBZ 8.8 Ki 2
NBVYRBDIADJELP 8.8 Ki 2
FPCBWBHSQIVWBN 8.8 Ki 3
KMKLFKWYYAVHDZ 8.8 Ki 3
PFSPMYHTZUFJQW 8.8 Ki 5
UWQNUCNXNKMWKG 8.8 Ki 5
ZJSWMRJWTWJORH 8.8 IC50 3
ITYRYCDVBXJIPH 8.8 IC50 2
LACTUOLELFMBLS 8.8 Ki 2
FJVQALKRJDSNIH 8.7 IC50 3
LIOWQNKZGLXNRL 8.7 IC50 3
VODYLGKYBHYDON 8.7 Ki 3
WCMVSMOIDILBOJ 8.7 Kd 5
ZPMRLGPLMNVIDC 8.7 Ki 4
ONSBLCCSCRKRKU 8.7 Ki 3
RTHXTYWCAPYZGF 8.7 Ki 3
GLRXSDVYMJTKAU 8.7 Ki 4
ITYRYCDVBXJIPH 8.7 IC50 2
KGGLWTNSVNKIRD 8.7 Ki 2
KVCMZPILKHYETB 8.7 Ki 2
UVVAXSWZJPKXLR 8.7 Ki 3
YKESQPGCPVQXIU 8.7 Ki 3
IEEFWRMSEALUNN 8.7 Kd 5
AKMDZGUFAAEGFX 8.7 Ki 5
FYYKZWOYOHYKPH 8.7 Ki 2
ZCGOYQXWRQDKNB 8.7 IC50 3
RKUNBYITZUJHSG 8.7 Ki 5
VKQLNHVNHKXWJD 8.7 Ki 2
WXIPHGJGJFDRNH 8.7 IC50 3
GLGYXEJECWKSPZ 8.6 Ki 3
QGACZOPMYZXVSJ 8.6 Ki 2
AVNRDCQRRUOTCC 8.6 Ki 5
BNLVIXOVYRJUTA 8.6 Ki 5
2D structure