Target Details
UniProt ACP08172
Gene SymbolCHRM2
Protein NameMuscarinic acetylcholine receptor M2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,645
  • Clinical molecules 27
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,645)
InChIKey pChEMBL Type Targets Clinical
NVEZMQGUUUDQFV 9.2 Ki 2
WFNJQDOBZMZPFU 9.2 Ki 2
ICZVKTVMHVHOQI 9.2 Ki 5
DDAFFKQDEBQDHP 9.1 Ki 3
DJOCICQNBMTMNG 9.1 Ki 5
MKNASJNZVVEVJG 9.1 Ki 2
SXLRCJRTHFTCEE 9.1 Ki 2
ZPUIFOBXUIMYGP 9.1 IC50 3
AZBTYTBTYGPQFW 9.1 Ki 2
LZCOQTDXKCNBEE 9.1 Ki 2
UUUTYZGDRKVSOB 9.1 Ki 2
WUMIJQZPHGJALC 9.1 Ki 2
ZGBSEJYQXDWFRF 9.1 Kd 2
JSDLJSSEKWSNAT 9.1 IC50 2
UCBXWLPRAVDTBU 9.1 Ki 5
WCMVSMOIDILBOJ 9.1 Ki 5
ZFXGEVATMHZGBZ 9.1 Ki 3
UBDKDGUJMUUUTQ 9.1 IC50 2
CBWGSRNEOFXWKO 9.1 IC50 3
VMJKUCKTXMESQR 9.1 Ki 5
GKNCQZVZUCNDGS 9.0 Ki 3
YXXULFOTUBYFOD 9.0 Ki 2
VLCYSUDIOLZSJK 9.0 Ki 3
ZYIJZBYORMBFMV 9.0 Ki 3
ZZCCWXNFFGHRJX 9.0 Ki 5
WCMVSMOIDILBOJ 9.0 Kd 5
DSYMOXJOJWZVRV 9.0 Ki 2
FLIWZNAGCZIAIW 9.0 Ki 2
MTYMLJSBEPCLGC 9.0 IC50 3
SIEQNGMENABBKP 9.0 Kd 3
SXLRCJRTHFTCEE 9.0 Ki 2
YQGXZPSEAUHNIN 9.0 Ki 4
ZGBSEJYQXDWFRF 9.0 Kd 2
OEXHQOGQTVQTAT 9.0 Ki 5
DFCLHAWGKPEFIX 9.0 Ki 5
ZMGKLIJUSAOHFP 9.0 IC50 3
DEFCMXPRFHURNR 9.0 Ki 2
JEEPGBSHIOBHQN 9.0 IC50 3
JGOIBENTSQHWDQ 9.0 Ki 5
OYYDSUSKLWTMMQ 8.9 Ki 5
UCURTLDVWIWPRM 8.9 Ki 5
XOZKVVSXDCLNPX 8.9 Ki 3
OEXHQOGQTVQTAT 8.9 Ki 5
VJOYACFUOINUHV 8.9 IC50 3
DIZOCNYCRPRXMN 8.9 Ki 3
GKNPSSNBBWDAGH 8.9 Ki 2
XTLIPTIWGCJFHQ 8.9 Kd 2
KWUNZCGOPMIGFE 8.9 IC50 2
OEXHQOGQTVQTAT 8.9 IC50 3
UBDKDGUJMUUUTQ 8.9 IC50 2
2D structure