Target Details
UniProt ACP08172
Gene SymbolCHRM2
Protein NameMuscarinic acetylcholine receptor M2
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 1,645
  • Clinical molecules 27
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,645)
InChIKey pChEMBL Type Targets Clinical
NGKTYFBTWFLIRS 9.5 Ki 4
SRLMLQNXERJQPS 9.5 Ki 4
XBBANBCTQDQYBC 9.5 Ki 4
JATHATTURQLZHF 9.5 Ki 2
YIMZVETVJULTMF 9.5 IC50 3
DLMOQVWYEFDOHH 9.4 Ki 5
IJOGXSLRDLSTOS 9.4 Ki 3
FRPQVLGDJMCCIJ 9.4 Ki 2
NBQAKYWBUGUZTQ 9.4 IC50 3
QRUXDRCXIGZTGT 9.4 Ki 5
REMJCBLKEGJHMN 9.4 IC50 3
BDWSAAGKPWOYAA 9.4 IC50 2
VBBBAIRVFNYIBU 9.4 Ki 2
BDZALISEBLHWIK 9.4 Ki 2
KLQQZEIBZUZRLW 9.4 Ki 4
LNNRXCJKYSSUPF 9.4 Ki 3
TWCNWISPABVKII 9.4 IC50 3
HGMITUYOCPPQLE 9.4 IC50 3
IECFFSCULPEXHT 9.4 Kd 3
LABGCBWSNGTBPM 9.4 Ki 2
YDKILWXULISVAK 9.4 Ki 2
DRCBVHVCMKPDSV 9.4 Ki 2
UFOTTYHVWBYOKX 9.4 Ki 5
LZCOQTDXKCNBEE 9.4 Ki 5
NVEZMQGUUUDQFV 9.4 IC50 3
GKNPSSNBBWDAGH 9.3 Ki 2
IJTZAYDMPFOINP 9.3 Ki 2
XXWOCVWJOICKHA 9.3 Kd 5
GPSZYYQYTBZUGG 9.3 IC50 3
KDMFWQZABCPNHX 9.3 Ki 2
AFLBGAQHDSOPKA 9.3 Ki 5
ROGWHWMEXSUERD 9.3 Ki 2
ANGKOCUUWGHLCE 9.3 IC50 5
KQHKTHFVDIBYJZ 9.3 IC50 5
RBDHPXXRYPWNOU 9.3 IC50 3
ZYZIHJMWCSZLEQ 9.3 IC50 3
BKJWZAJINPBJAC 9.2 Ki 2
FNAJWFJEAUHFJC 9.2 Ki 2
FYYWKHFZJYSOCA 9.2 IC50 2
YFWMVRIRFFWDJL 9.2 Ki 5
AWMYFVQONDTWPK 9.2 Ki 2
CFPVEUFKLQKJRS 9.2 IC50 3
CZMLHCKAVIBNFO 9.2 Ki 2
LLPYCIXHQOFZRV 9.2 IC50 3
XJFLDBYRKJAMIK 9.2 Kd 5
QJBDLOQOXGQJTD 9.2 Ki 5
QOXJSXPGWIRRNX 9.2 Ki 5
NHUURXLCGOCXHZ 9.2 IC50 5
KFMIEAZKENMLEL 9.2 Kd 5
CWHBWBZGFMIKAF 9.2 Ki 3
2D structure