Target Details
| UniProt AC | P08069 |
|---|---|
| Gene Symbol | IGF1R |
| Protein Name | Insulin-like growth factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 611
- Clinical molecules 120
- Avg pChEMBL 7.78
KEGG Pathways (32)
- AMPK signaling pathway
- Adherens junction
- Autophagy - animal
- Breast cancer
- Cadherin signaling
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Focal adhesion
- FoxO signaling pathway
- Glioma
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Hormone signaling
- Integrin signaling
- Long-term depression
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Melanoma
- Oocyte meiosis
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Signaling pathways regulating pluripotency of stem cells
- Transcriptional misregulation in cancer
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (611)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AHPTUXAIRHFFGA
|
7.0 | IC50 | 2 | — | |
ASBGJVNBZBSENK
|
7.0 | IC50 | 2 | — | |
CQFVDHNTTRWVQD
|
7.0 | Ki | 9 | — | |
FTKTXHIRMKWXBE
|
7.0 | IC50 | 2 | — | |
GQGMUKOYILWOIQ
|
7.0 | Ki | 25 | — | |
JGMJCQJURLCLJC
|
7.0 | IC50 | 2 | — | |
KUYIQVZTFYAICK
|
7.0 | IC50 | 2 | — | |
LAVUQVGESJYCJA
|
7.0 | IC50 | 2 | — | |
LQZVTJLMRRUWTJ
|
7.0 | IC50 | 5 | Yes | |
NQBOWNPIRYVPJI
|
7.0 | IC50 | 2 | — | |
OCTJJTONFVZCDV
|
7.0 | IC50 | 2 | — | |
QSNLBMCGRQUEPH
|
7.0 | IC50 | 2 | — | |
RNICSIBFPJOYHB
|
7.0 | IC50 | 2 | — | |
UOUIRSAMKHDQKN
|
7.0 | IC50 | 2 | — | |
UUFDRURWKKKAJF
|
7.0 | IC50 | 4 | Yes | |
VKBFHTIUXUCYRQ
|
7.0 | Ki | 66 | — | |
XRMQCRQMFWASRC
|
7.0 | IC50 | 2 | — | |
YRUIXESBPXQWOD
|
7.0 | IC50 | 3 | — | |
ZQOJOCBLMULSIQ
|
7.0 | IC50 | 3 | — | |
ZWVZORIKUNOTCS
|
7.0 | IC50 | 10 | Yes | |
RJTVPQLMBWIFKC
|
7.0 | IC50 | 5 | — | |
NXVHOYBQFPQTBF
|
7.0 | Ki | 3 | — | |
LDLBFITVAGVRNV
|
7.0 | IC50 | 6 | Yes | |
YBJHTHAFJHFCAF
|
7.0 | IC50 | 3 | Yes | |
SSPYHBZSDDTSFN
|
7.0 | IC50 | 9 | — | |
UAKYYEQJRKJUBT
|
7.0 | Ki | 5 | Yes | |
HKJUUPKKOAGVDB
|
6.9 | IC50 | 6 | Yes | |
HKSZLNNOFSGOKW
|
6.9 | IC50 | 408 | — | |
LDRVTAIULYJYRP
|
6.9 | IC50 | 2 | — | |
RZNBLEUQXRTRGF
|
6.9 | IC50 | 2 | — | |
COPINYWCESNOFK
|
6.9 | IC50 | 3 | — | |
COPINYWCESNOFK
|
6.9 | IC50 | 3 | — | |
PSLCBMWJMHKRLT
|
6.9 | IC50 | 3 | Yes | |
VJWLMBVALMQEMA
|
6.9 | IC50 | 3 | — | |
ZTKZGNHMDMISHE
|
6.9 | IC50 | 3 | — | |
DPQSQXGBMAXUAP
|
6.9 | IC50 | 3 | — | |
BLGAPWCYLDPMFH
|
6.9 | IC50 | 2 | — | |
SZCXARSUVUOVCP
|
6.9 | IC50 | 3 | — | |
XKZQZMSAWVDRSP
|
6.8 | IC50 | 39 | Yes | |
ZTSJUQOBFLZJMJ
|
6.8 | IC50 | 2 | — | |
FIODPWXACNUFML
|
6.8 | Ki | 2 | — | |
HBAGNJCIEGUKLI
|
6.8 | IC50 | 2 | — | |
LDRHWDNTNFXKEE
|
6.8 | Ki | 3 | — | |
XTPHJLPNQUXWCD
|
6.8 | Ki | 3 | — | |
FILMJNHPVCSZTN
|
6.8 | IC50 | 2 | — | |
MJEHBQIPZHTMNZ
|
6.8 | IC50 | 2 | — | |
MNMQBQOLMHVBJT
|
6.8 | Ki | 3 | Yes | |
OCNLJCSEDBMGNF
|
6.8 | IC50 | 2 | — | |
BCCBBFDXEPUOFF
|
6.8 | IC50 | 3 | Yes | |
CZVVMRNEBRFYTL
|
6.8 | IC50 | 9 | Yes |