Target Details
| UniProt AC | P08069 |
|---|---|
| Gene Symbol | IGF1R |
| Protein Name | Insulin-like growth factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 611
- Clinical molecules 120
- Avg pChEMBL 7.78
KEGG Pathways (32)
- AMPK signaling pathway
- Adherens junction
- Autophagy - animal
- Breast cancer
- Cadherin signaling
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Focal adhesion
- FoxO signaling pathway
- Glioma
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Hormone signaling
- Integrin signaling
- Long-term depression
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Melanoma
- Oocyte meiosis
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Signaling pathways regulating pluripotency of stem cells
- Transcriptional misregulation in cancer
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (611)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UEBUEWAMMXNGMS
|
7.3 | IC50 | 2 | — | |
WLEKHBHSQHEZQU
|
7.3 | IC50 | 2 | Yes | |
JUSBGYZKUCMHQQ
|
7.3 | IC50 | 2 | — | |
XIQAFZIFYBEQQW
|
7.3 | IC50 | 3 | — | |
ZJDFSKSBQBPOSK
|
7.3 | IC50 | 24 | Yes | |
DEBFWFAAIWZWSH
|
7.3 | IC50 | 3 | — | |
WDRXGELIQZMTRU
|
7.3 | IC50 | 3 | — | |
ONDLPAJKNFWPJO
|
7.3 | IC50 | 2 | — | |
BPFRWNTWHHVPFL
|
7.2 | IC50 | 2 | — | |
MOSKATHMXWSZTQ
|
7.2 | IC50 | 16 | Yes | |
VERWOWGGCGHDQE
|
7.2 | IC50 | 23 | — | |
ZAKBVBOEYCRZJE
|
7.2 | IC50 | 2 | — | |
GERKWUCMHZITIS
|
7.2 | IC50 | 2 | — | |
KKACLEOGRMSWFM
|
7.2 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.2 | Kd | 165 | Yes | |
ZUXJDKZUOTZPMQ
|
7.2 | IC50 | 2 | Yes | |
AECDBHGVIIRMOI
|
7.2 | IC50 | 7 | — | |
MSLPPMUTXCBVLE
|
7.2 | IC50 | 4 | Yes | |
HXLFOHIDCPNVHE
|
7.2 | IC50 | 3 | Yes | |
QSENMPAGYMUVDE
|
7.2 | IC50 | 5 | — | |
SLFIVXXZOYCJGB
|
7.2 | IC50 | 3 | — | |
FHQQNAHMJMQUKJ
|
7.2 | IC50 | 4 | Yes | |
NWGRWOHGDXCBOV
|
7.2 | IC50 | 4 | Yes | |
VZGOJYYBQQYRJE
|
7.2 | IC50 | 2 | — | |
DPDFZTKJHYCDSX
|
7.2 | Ki | 3 | — | |
MHAJGINRQAEMIM
|
7.1 | IC50 | 2 | — | |
SGQJPPQXKVUHGS
|
7.1 | IC50 | 6 | Yes | |
SKBWQUPLWQUWPH
|
7.1 | IC50 | 6 | Yes | |
OQEBLEZRSCIFJK
|
7.1 | IC50 | 2 | — | |
DLQXAWIVHRHOQT
|
7.1 | IC50 | 6 | Yes | |
MQCNUAFNUAISQK
|
7.1 | IC50 | 3 | — | |
SRUYMJRFVGLQDV
|
7.1 | Ki | 37 | — | |
TVUWQDLBEOZVOU
|
7.1 | Ki | 41 | — | |
UYHKCQAFCWYUAF
|
7.1 | IC50 | 2 | — | |
DRQNCWQLZYUQOI
|
7.1 | IC50 | 2 | — | |
JHZWEYCWMPNVEC
|
7.1 | IC50 | 4 | Yes | |
MFPBQNCVIIGPOV
|
7.1 | IC50 | 4 | Yes | |
OBDZFXLPCBGQSA
|
7.1 | IC50 | 3 | — | |
UETYAVAIGWIDEO
|
7.1 | IC50 | 3 | — | |
UYJNQQDJUOUFQJ
|
7.1 | IC50 | 68 | — | |
YETDQFJRLHRQJD
|
7.1 | IC50 | 4 | Yes | |
ZRTDGPKHIJCQNA
|
7.1 | IC50 | 3 | — | |
USVCWSAJUAARAL
|
7.1 | IC50 | 8 | — | |
DMUUMPYJFUHKCR
|
7.1 | Ki | 2 | — | |
FBFCEASGGVTKEY
|
7.1 | IC50 | 6 | — | |
LZNLVKVRHVELDP
|
7.1 | IC50 | 3 | — | |
YHAJJCOJWJKFSB
|
7.1 | IC50 | 2 | — | |
CGJRRFJDMMUHJW
|
7.0 | IC50 | 5 | Yes | |
JZMKNOWKNYJUOM
|
7.0 | Ki | 3 | — | |
YUEGRPWDOBJWDW
|
7.0 | IC50 | 3 | — |