Target Details
| UniProt AC | P08069 |
|---|---|
| Gene Symbol | IGF1R |
| Protein Name | Insulin-like growth factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 611
- Clinical molecules 120
- Avg pChEMBL 7.78
KEGG Pathways (32)
- AMPK signaling pathway
- Adherens junction
- Autophagy - animal
- Breast cancer
- Cadherin signaling
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Focal adhesion
- FoxO signaling pathway
- Glioma
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Hormone signaling
- Integrin signaling
- Long-term depression
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Melanoma
- Oocyte meiosis
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Signaling pathways regulating pluripotency of stem cells
- Transcriptional misregulation in cancer
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (611)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YXLQJZQRBVGUCM
|
7.9 | IC50 | 2 | — | |
ZNLCRBCFRLCIFE
|
7.9 | IC50 | 4 | Yes | |
ILKQWXHVEJRPAL
|
7.8 | IC50 | 2 | — | |
RTGPQVHYQAWJEV
|
7.8 | IC50 | 2 | — | |
SIVMXJQFCAHOMI
|
7.8 | IC50 | 2 | — | |
KJDKBIYPTUYYHT
|
7.8 | IC50 | 2 | — | |
PXCKFKLPESDHTQ
|
7.8 | IC50 | 2 | — | |
BOJLJYRVWHJBLQ
|
7.8 | IC50 | 2 | — | |
MKEZXJZAKPJGKM
|
7.8 | IC50 | 2 | — | |
SCJMHNYQTKWNRD
|
7.8 | IC50 | 2 | — | |
RQDNRYSBNFWQCV
|
7.8 | IC50 | 3 | — | |
SBLMCLDRWJNEJK
|
7.7 | IC50 | 17 | — | |
QPKFJNSFZBUDOA
|
7.7 | Ki | 2 | — | |
FUGZYLOFWXVFQU
|
7.7 | IC50 | 3 | Yes | |
KJWZHCRQZUOQJR
|
7.7 | IC50 | 3 | — | |
KZKWIMSZKNQYFJ
|
7.7 | IC50 | 2 | — | |
YHWJHUBPWLCING
|
7.7 | IC50 | 3 | — | |
FYSLYZBOZFMTDD
|
7.7 | IC50 | 6 | Yes | |
IBXPUECEDDUZFG
|
7.7 | IC50 | 3 | — | |
PKCDDUHJAFVJJB
|
7.7 | IC50 | 13 | — | |
CAXBBGZEJPMNQW
|
7.6 | IC50 | 2 | — | |
CFIBXVQLBVNOHW
|
7.6 | Ki | 64 | — | |
CZRPHLYGJSYQCK
|
7.6 | IC50 | 2 | Yes | |
FLEAYYMORDPWAJ
|
7.6 | Ki | 90 | — | |
FNIODIAGYLWZRY
|
7.6 | IC50 | 4 | Yes | |
GGQTUXCKDZGJDL
|
7.6 | IC50 | 2 | Yes | |
ILUGAYBMBIJXHC
|
7.6 | Ki | 9 | — | |
OSHPEWCCDRPGGK
|
7.6 | Ki | 3 | — | |
YEHCNYAQEBQCCS
|
7.6 | Ki | 74 | — | |
ZWVZORIKUNOTCS
|
7.6 | Ki | 69 | — | |
MWTCMQXTURNBFI
|
7.6 | IC50 | 4 | Yes | |
PZKWAHCUWGHBLH
|
7.6 | IC50 | 7 | — | |
RDFZVFFSXWGAKR
|
7.6 | IC50 | 2 | — | |
RFZOHHKCEHQQBE
|
7.6 | IC50 | 3 | — | |
UMWXVGCBUMYAFH
|
7.6 | Ki | 3 | — | |
AIDASDNWZFQVSE
|
7.6 | Ki | 2 | — | |
CCVGHLZQHJYDAI
|
7.6 | IC50 | 3 | — | |
FXYPQFBJRKMLDS
|
7.6 | IC50 | 4 | — | |
JKKIQRNCGVRLBH
|
7.6 | IC50 | 2 | — | |
JNGUPQQSJDYXDB
|
7.6 | IC50 | 2 | — | |
PXOJXTKZVIEYLV
|
7.6 | IC50 | 4 | Yes | |
UMHKPLNSKRNIJU
|
7.6 | IC50 | 2 | — | |
VWCZORWQNKCYGE
|
7.6 | IC50 | 17 | — | |
SKXAZUOZHANICG
|
7.5 | IC50 | 3 | — | |
UXGODHMBZZMTNL
|
7.5 | IC50 | 2 | — | |
ZJATUHGFXPEBQJ
|
7.5 | IC50 | 2 | — | |
LVOHHKIFPDWJJY
|
7.5 | IC50 | 2 | — | |
LVOHHKIFPDWJJY
|
7.5 | IC50 | 2 | — | |
MFFQPYYPGSJIDM
|
7.5 | IC50 | 2 | — | |
PDJARQSWGDDFHH
|
7.5 | IC50 | 4 | — |