Target Details
| UniProt AC | P08069 |
|---|---|
| Gene Symbol | IGF1R |
| Protein Name | Insulin-like growth factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 611
- Clinical molecules 120
- Avg pChEMBL 7.78
KEGG Pathways (32)
- AMPK signaling pathway
- Adherens junction
- Autophagy - animal
- Breast cancer
- Cadherin signaling
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Focal adhesion
- FoxO signaling pathway
- Glioma
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Hormone signaling
- Integrin signaling
- Long-term depression
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Melanoma
- Oocyte meiosis
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Signaling pathways regulating pluripotency of stem cells
- Transcriptional misregulation in cancer
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (611)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IILFQZAVZNEIKL
|
9.0 | IC50 | 2 | — | |
JFJRYQOFIDFJKY
|
9.0 | IC50 | 2 | Yes | |
JKGUWRSWKIHSTP
|
9.0 | IC50 | 2 | — | |
KCFKHBXTNWBJGZ
|
9.0 | IC50 | 2 | — | |
KCZLTVJTTQQVRB
|
9.0 | IC50 | 2 | — | |
LUUOHJCBIJQUBZ
|
9.0 | IC50 | 2 | — | |
MAYBCHWSKBRUDW
|
9.0 | IC50 | 2 | — | |
NACGODPXQGEECG
|
9.0 | IC50 | 2 | Yes | |
OTTBPQUZNFGLAM
|
9.0 | IC50 | 2 | Yes | |
QUMKTRJRHYFANK
|
9.0 | IC50 | 2 | Yes | |
RXYPFHYDNNLDSN
|
9.0 | IC50 | 2 | — | |
RKXGEBJVNGSICG
|
8.9 | IC50 | 3 | — | |
DGIKQZFVNNRZMT
|
8.8 | IC50 | 3 | — | |
CGLNKCUZVMEOBR
|
8.8 | IC50 | 3 | Yes | |
USFRNJSCBVCBFY
|
8.8 | IC50 | 4 | Yes | |
FLTJPMCKNUNPRH
|
8.8 | IC50 | 3 | — | |
BHLTVGNUTOSHBD
|
8.7 | IC50 | 3 | — | |
WDUXPXHDIYWLHP
|
8.7 | IC50 | 3 | — | |
ASLJKKCVGZGUQJ
|
8.7 | IC50 | 3 | Yes | |
AUQYWFVTSGUQCD
|
8.7 | IC50 | 2 | — | |
GBWMNCWACPCEEQ
|
8.7 | IC50 | 2 | — | |
HFMMOXFTBXCGCO
|
8.7 | IC50 | 2 | — | |
HJERFKFVQHRAML
|
8.7 | IC50 | 2 | — | |
HXZDICYKFAOZLE
|
8.7 | IC50 | 6 | Yes | |
KXWPCIASWBFLMB
|
8.7 | IC50 | 2 | — | |
MZVQVCMUWUQNFP
|
8.7 | IC50 | 2 | — | |
ODJRLLIFPOKNLG
|
8.7 | IC50 | 2 | — | |
OJOAXIFFWKGMCG
|
8.7 | IC50 | 2 | — | |
POARIJJCCJDSKV
|
8.7 | IC50 | 5 | Yes | |
SOSWXMRNLZWISK
|
8.7 | IC50 | 3 | — | |
WHVFDYQCAMPLMS
|
8.7 | IC50 | 20 | Yes | |
WMNYFCPOALWAPO
|
8.7 | IC50 | 2 | Yes | |
YPPZOXGKXXTCAP
|
8.7 | IC50 | 2 | — | |
YRONGIKDOAUNNP
|
8.7 | IC50 | 2 | — | |
YUIOENQMCZQWAY
|
8.7 | IC50 | 2 | — | |
ZBUFIMGFTPZODR
|
8.7 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
8.7 | IC50 | 33 | Yes | |
YSRFTZRNFJRVPH
|
8.6 | IC50 | 5 | Yes | |
QQWUGDVOUVUTOY
|
8.6 | IC50 | 231 | Yes | |
BYCKMIYPESNKTL
|
8.5 | IC50 | 2 | Yes | |
CJLMCBMDZOAJLV
|
8.5 | IC50 | 2 | — | |
FJMVOCSRTVXRIV
|
8.5 | IC50 | 2 | — | |
IBDMRAZGYXXBKY
|
8.5 | IC50 | 2 | — | |
KUQOZTZPJMJBMT
|
8.5 | IC50 | 3 | — | |
PLCWQDVCBVWDJZ
|
8.5 | IC50 | 2 | — | |
OVDSPTSBIQCAIN
|
8.5 | IC50 | 7 | — | |
KTQGBACJIGNCAB
|
8.4 | IC50 | 3 | — | |
CDXYAHJJGRNDCW
|
8.4 | IC50 | 3 | Yes | |
CGMDMXYNDLBSNT
|
8.4 | IC50 | 5 | Yes | |
IKALKYJLFRWHAR
|
8.4 | IC50 | 2 | — |