Target Details
| UniProt AC | P08069 |
|---|---|
| Gene Symbol | IGF1R |
| Protein Name | Insulin-like growth factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 611
- Clinical molecules 120
- Avg pChEMBL 7.78
KEGG Pathways (32)
- AMPK signaling pathway
- Adherens junction
- Autophagy - animal
- Breast cancer
- Cadherin signaling
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Focal adhesion
- FoxO signaling pathway
- Glioma
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Hormone signaling
- Integrin signaling
- Long-term depression
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Melanoma
- Oocyte meiosis
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Signaling pathways regulating pluripotency of stem cells
- Transcriptional misregulation in cancer
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (611)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JCAOTPBZOINVCN
|
9.4 | IC50 | 2 | — | |
LWVQAFSEKOOOAI
|
9.4 | IC50 | 2 | — | |
OPSIJGYSVYFFGS
|
9.4 | IC50 | 2 | — | |
OYQMWWVIYBSJLB
|
9.4 | IC50 | 2 | — | |
UVJDZKBPVPTIRA
|
9.4 | IC50 | 2 | — | |
YRLINYQMYNEFJG
|
9.4 | IC50 | 2 | — | |
GLSBPQXKUMSIMB
|
9.4 | IC50 | 2 | — | |
HUHCYTMKDOFWSG
|
9.4 | IC50 | 2 | — | |
LDYDMNAZFRCWNR
|
9.4 | IC50 | 2 | — | |
RKWGNTHTPQXXQN
|
9.4 | IC50 | 2 | — | |
RZLRBIAISAXDHA
|
9.4 | IC50 | 2 | — | |
HFTHUIUDNIONGS
|
9.4 | IC50 | 3 | — | |
QJWZXYIVWQUAAO
|
9.4 | IC50 | 2 | — | |
KVFQSNCDMQJZPD
|
9.4 | IC50 | 2 | — | |
IQLMHUMYHUUAQQ
|
9.4 | IC50 | 2 | — | |
JGLSPBGRSLPKAQ
|
9.3 | IC50 | 2 | — | |
QJSZKBYCIGDBBS
|
9.3 | IC50 | 2 | — | |
LEVAPGLCIYCDDH
|
9.3 | IC50 | 3 | — | |
FHMWNSNIIZHZPJ
|
9.3 | IC50 | 2 | — | |
PTPQXKBVULYOLN
|
9.3 | IC50 | 2 | — | |
IAIFZADOAVHXEL
|
9.3 | IC50 | 2 | — | |
IKWHWJFNGWUVIJ
|
9.3 | IC50 | 2 | Yes | |
MUAJURKWULOSJG
|
9.3 | IC50 | 2 | — | |
ZZJJJCFYECEHNN
|
9.3 | IC50 | 2 | — | |
CWSQJENYIZLGER
|
9.3 | IC50 | 2 | — | |
YDCSUBLUYMXIOG
|
9.2 | IC50 | 2 | — | |
NXJDOMZWUPMZFE
|
9.2 | IC50 | 2 | — | |
RVIMGPNKJMIZJW
|
9.2 | IC50 | 2 | — | |
RNRVBUQQZHOCBU
|
9.2 | IC50 | 2 | — | |
BHOLGBKCKRPFPA
|
9.2 | IC50 | 2 | — | |
GWVCRFPHEQXQJR
|
9.2 | IC50 | 2 | — | |
DMQJVMSMJXCZOS
|
9.2 | IC50 | 2 | — | |
ALHWHMNSEAIFMC
|
9.2 | IC50 | 2 | — | |
YEPYKAAAXUCSMP
|
9.1 | IC50 | 2 | — | |
QWPNPMFVZNBPEA
|
9.1 | IC50 | 2 | — | |
VVXWJQWOEIYIHP
|
9.1 | IC50 | 2 | — | |
ZCTVEBRXLFXVIK
|
9.1 | IC50 | 3 | — | |
VZVLZJITGHRMBT
|
9.1 | IC50 | 2 | — | |
BAIRSNTWXBQKHG
|
9.1 | IC50 | 2 | — | |
PCUMDMKSEZJNLA
|
9.1 | IC50 | 2 | — | |
ZSIGECCEZMACTJ
|
9.1 | IC50 | 2 | — | |
YQWFNFUEJRELJX
|
9.1 | IC50 | 2 | — | |
CZHQIACJGGUSQU
|
9.1 | IC50 | 2 | — | |
DLKUDUSWHQNMDW
|
9.1 | IC50 | 2 | — | |
SBDSSXKUILJHSM
|
9.1 | IC50 | 2 | — | |
LGLJGJQDMXPFHU
|
9.0 | IC50 | 2 | — | |
SFBCVPDTLHGKAL
|
9.0 | IC50 | 2 | — | |
DUOSEXDXCYSSSZ
|
9.0 | IC50 | 2 | Yes | |
FENCVPRSVOEMHI
|
9.0 | IC50 | 2 | — | |
GHPFQRTVUDXWCC
|
9.0 | Ki | 35 | — |