Target Details
| UniProt AC | P08069 |
|---|---|
| Gene Symbol | IGF1R |
| Protein Name | Insulin-like growth factor 1 receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00757 (Furin-like) PF07714 (PK_Tyr_Ser-Thr) PF01030 (Recep_L_domain) |
Summary
- Multi-target molecules 611
- Clinical molecules 120
- Avg pChEMBL 7.78
KEGG Pathways (32)
- AMPK signaling pathway
- Adherens junction
- Autophagy - animal
- Breast cancer
- Cadherin signaling
- EGFR tyrosine kinase inhibitor resistance
- Endocrine resistance
- Endocytosis
- Focal adhesion
- FoxO signaling pathway
- Glioma
- HIF-1 signaling pathway
- Hepatocellular carcinoma
- Hormone signaling
- Integrin signaling
- Long-term depression
- Longevity regulating pathway
- Longevity regulating pathway - multiple species
- MAPK signaling pathway
- Melanoma
- Oocyte meiosis
- Ovarian steroidogenesis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Progesterone-mediated oocyte maturation
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Signaling pathways regulating pluripotency of stem cells
- Transcriptional misregulation in cancer
- mTOR signaling pathway
Associated Diseases (4)
Active Molecules (611)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DWLZYJOAPBAXQM
|
10.3 | IC50 | 2 | — | |
FLBQTCODPBJFTD
|
10.3 | IC50 | 2 | — | |
DANRHRCSZZGXLP
|
10.1 | IC50 | 2 | — | |
KUXYUFHYERAGDG
|
10.1 | IC50 | 2 | — | |
WFXSEBKHQBTMMS
|
10.1 | IC50 | 2 | — | |
ZEPVDOIWFVBKOM
|
10.1 | IC50 | 2 | — | |
GBTTYDWBVFNAEA
|
10.1 | IC50 | 2 | — | |
MRNCAMTZMKCLDO
|
10.1 | IC50 | 2 | — | |
NWCSJPOCTCBOEW
|
10.1 | IC50 | 2 | — | |
DKWOGWIUVLBDHC
|
10.0 | IC50 | 2 | — | |
DRYYTRLZCKWIGZ
|
10.0 | IC50 | 2 | — | |
KZXBXGNMGTZACU
|
10.0 | IC50 | 2 | — | |
URABRDOUNMLPLA
|
10.0 | IC50 | 2 | — | |
KXDLJCXLOFTQOJ
|
10.0 | IC50 | 2 | — | |
SOUDXNZKWYTFFW
|
10.0 | IC50 | 2 | — | |
XRVFEWYOEIYZGB
|
10.0 | IC50 | 3 | — | |
PAEPNROAXKXFOQ
|
9.9 | IC50 | 2 | — | |
JRKWDAZGBOBRPT
|
9.9 | IC50 | 2 | — | |
MRTQXPYBEKCXAN
|
9.9 | IC50 | 2 | — | |
MZRCFUHXHKAGCK
|
9.9 | IC50 | 2 | — | |
NJBNQVCQKINYLS
|
9.9 | IC50 | 2 | — | |
OWPFZNYKPFPFIT
|
9.9 | IC50 | 2 | — | |
YOFGUEQIPVDBEL
|
9.9 | IC50 | 2 | — | |
GLLLAYKUVMFJER
|
9.8 | IC50 | 2 | — | |
GMHBLFNISBWXBO
|
9.8 | IC50 | 2 | — | |
SDTDXGMQPJHODR
|
9.8 | IC50 | 2 | — | |
WSEOWNBBPGNYRJ
|
9.8 | IC50 | 2 | — | |
XYBRNZWRDMIYFT
|
9.8 | IC50 | 2 | — | |
BKYSHTIOCHNDDH
|
9.8 | IC50 | 2 | — | |
CNBMRJSFULHWLZ
|
9.8 | IC50 | 2 | — | |
FCGZIEABISYQOO
|
9.8 | IC50 | 2 | — | |
CLXCUJAIQNKPCW
|
9.8 | IC50 | 2 | — | |
DEUXRKZJLFSYAO
|
9.8 | IC50 | 2 | — | |
IYYUJNJRKWXTJJ
|
9.8 | IC50 | 2 | — | |
NDVDUHONBQZAGA
|
9.8 | IC50 | 2 | — | |
OSGQGIINHNRMCL
|
9.8 | IC50 | 2 | — | |
RXLGVLBKICWANA
|
9.8 | IC50 | 2 | — | |
SAJTWQRLZVYSCP
|
9.8 | IC50 | 2 | — | |
UHHADNYIBMJTNI
|
9.8 | IC50 | 2 | — | |
VJSMYRLRQBWBQP
|
9.8 | IC50 | 2 | — | |
HCMFOVBYPFSDST
|
9.8 | IC50 | 2 | — | |
IEFXGIIDRDRIGF
|
9.8 | IC50 | 2 | — | |
IEMCBHBTNFUENC
|
9.8 | IC50 | 2 | — | |
OPYZOEXGCQPJNO
|
9.8 | IC50 | 2 | — | |
RWSCTJGHFHKJNJ
|
9.8 | IC50 | 2 | — | |
IBFTXGLRFZFDGT
|
9.7 | IC50 | 2 | — | |
IDUFXVFDCDFZDE
|
9.7 | IC50 | 2 | — | |
QSOSQIVFCJZEIL
|
9.7 | IC50 | 2 | — | |
UBDSRPCDONKGEF
|
9.7 | IC50 | 2 | — | |
DXLDXBDJHXQCCM
|
9.7 | IC50 | 2 | — |