Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XHZDAKAAKUZJHY
|
7.2 | IC50 | 4 | — | |
ATYKMHIJRBRZOA
|
7.2 | IC50 | 2 | — | |
LROXDAJCTUTCNN
|
7.2 | IC50 | 2 | — | |
BLQYVHBZHAISJM
|
7.2 | IC50 | 21 | Yes | |
FWXNEFMIRVAQLN
|
7.1 | IC50 | 4 | — | |
OKHZIVXQKINVAO
|
7.1 | IC50 | 4 | — | |
ARRUJZPOJKKPKY
|
7.1 | IC50 | 3 | — | |
BKDBTNDUTIFYHL
|
7.1 | IC50 | 2 | — | |
CNYOFMNBFMTOHX
|
7.1 | IC50 | 5 | — | |
JOOXLOJCABQBSG
|
7.1 | Kd | 139 | — | |
BYVUAJDYENVNAV
|
7.1 | IC50 | 3 | — | |
FWQLGWJRPGEROE
|
7.1 | Ki | 2 | — | |
JZTOUVBEZONDKA
|
7.1 | Ki | 80 | — | |
MTCHQDWUHQADSY
|
7.1 | Ki | 29 | — | |
QZKXRJMVQTZACR
|
7.1 | IC50 | 3 | — | |
RAPYFGJGASETOS
|
7.1 | Ki | 11 | — | |
RTDSHUGNRVXRHN
|
7.1 | Ki | 51 | — | |
RYAVJHIPOWNWDE
|
7.1 | Ki | 38 | — | |
SBWCIJOOABLPME
|
7.1 | Ki | 13 | — | |
YMIJUBCSOKSFRU
|
7.1 | Ki | 87 | — | |
ZVWRFVCNQOECJS
|
7.1 | Ki | 71 | — | |
FNKZXYIORCSWOH
|
7.1 | IC50 | 2 | — | |
OSAWFUCUZJNEID
|
7.0 | IC50 | 20 | — | |
GZPJCJKUZPUFAL
|
7.0 | Kd | 4 | — | |
CEQUQTKEVIQAMX
|
7.0 | IC50 | 3 | — | |
OIANGKGOYKDGQV
|
7.0 | Kd | 10 | — | |
YZNIHXUBUWEUCM
|
7.0 | IC50 | 14 | — | |
HCNIBOQWDVOZKF
|
7.0 | Ki | 26 | — | |
KXPWWMPXNUOYOH
|
7.0 | Ki | 24 | — | |
LCGSWTFWYNYUKS
|
7.0 | Ki | 26 | — | |
LRLDYTTWQIFWBD
|
7.0 | Ki | 25 | — | |
NMJIPDOHEVXEHN
|
7.0 | IC50 | 3 | — | |
SEVCBWKJSOLMNQ
|
7.0 | Ki | 38 | — | |
SPMHGQZFMNZCBV
|
7.0 | Ki | 30 | Yes | |
TXHOCWWJSGCZLC
|
7.0 | Ki | 18 | — | |
VHFBRSZCMAZULY
|
7.0 | IC50 | 2 | — | |
VQPBIJGXSXEOCU
|
7.0 | Ki | 24 | — | |
YDOPLCNFRXOHCC
|
7.0 | Ki | 28 | — | |
RITAVMQDGBJQJZ
|
7.0 | Kd | 43 | — | |
CIVSWNZKBWESRB
|
7.0 | IC50 | 6 | — | |
TVJRDCQUZMGBAB
|
7.0 | IC50 | 13 | — | |
URLYPAWCHVXIAA
|
7.0 | IC50 | 4 | Yes | |
WKDACQVEJIVHMZ
|
7.0 | Kd | 46 | — | |
WPEWQEMJFLWMLV
|
7.0 | Kd | 2 | — | |
XYHJHIRTHHPPSJ
|
7.0 | IC50 | 2 | — | |
GBJVVSCPOBPEIT
|
7.0 | Kd | 13 | Yes | |
ORWIYCURPDKSBI
|
7.0 | IC50 | 15 | Yes | |
YABJJWZLRMPFSI
|
6.9 | Kd | 34 | — | |
MPVGZUGXCQEXTM
|
6.9 | Kd | 61 | Yes | |
QYZOGCMHVIGURT
|
6.9 | Kd | 26 | Yes |