Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KSCKIOGOWXGQCD
|
7.3 | IC50 | 2 | — | |
QHXBWJSQXSYAGG
|
7.3 | IC50 | 16 | — | |
JUIHREVFVXLZPR
|
7.3 | IC50 | 10 | — | |
PIQCTGMSNWUMAF
|
7.3 | Kd | 137 | Yes | |
YYLKKYCXAOBSRM
|
7.3 | Kd | 191 | — | |
XRFFUVUJIBWJII
|
7.3 | IC50 | 3 | — | |
BSFNGHCTZDCQBF
|
7.3 | Ki | 93 | — | |
GMYYMEOGFRKSFS
|
7.3 | Ki | 29 | — | |
HEUSUIRCBWROMH
|
7.3 | Ki | 64 | — | |
KOHNRDPXFDZZJF
|
7.3 | Ki | 31 | — | |
MMJWZGGVKOHMPQ
|
7.3 | IC50 | 6 | — | |
NXNQLECPAXXYTR
|
7.3 | Ki | 29 | — | |
OGNYUTNQZVRGMN
|
7.3 | Ki | 16 | Yes | |
QXRJBJVCBQSLTA
|
7.3 | Ki | 29 | — | |
RGNHKJWHFIPHIM
|
7.3 | Ki | 66 | — | |
UWDBNTXEKYRMSG
|
7.3 | Ki | 26 | — | |
XLFYOIVELARSKP
|
7.3 | Ki | 33 | — | |
MPKFPGZSQMILTQ
|
7.3 | IC50 | 5 | — | |
OSVUGUHRKMMBSE
|
7.3 | Kd | 170 | — | |
XCJXNMGPLVXHMC
|
7.3 | IC50 | 4 | — | |
JQOIRTDBHMDWMT
|
7.3 | IC50 | 2 | — | |
NDEXUOWTGYUVGA
|
7.3 | IC50 | 12 | — | |
ZHOXAGNPCZTRBN
|
7.3 | Kd | 20 | — | |
SRQQRYTWWRXHKL
|
7.2 | IC50 | 2 | — | |
ZHPRBIFEDSMSRL
|
7.2 | IC50 | 2 | — | |
JROFGZPOBKIAEW
|
7.2 | Kd | 10 | — | |
KOFXELGVKHKUJR
|
7.2 | IC50 | 3 | — | |
UGPDJIJFANODJH
|
7.2 | IC50 | 12 | — | |
VAARYSWULJUGST
|
7.2 | Kd | 119 | Yes | |
OYIGMLCBXUNGGL
|
7.2 | IC50 | 3 | — | |
ACNCCUVYXQGPKZ
|
7.2 | Ki | 31 | — | |
DOLVPVSWTLFZMQ
|
7.2 | Ki | 17 | — | |
GCBJDOWIQHMCMR
|
7.2 | Ki | 84 | — | |
HDWGWERBFXSKLX
|
7.2 | IC50 | 2 | — | |
KEZAHTDTAWUZDU
|
7.2 | Ki | 8 | — | |
KRIUNPBAQZGFQA
|
7.2 | Ki | 76 | — | |
LYNBNVBMAGDJRW
|
7.2 | Ki | 81 | — | |
MADCXGNPDBWPLM
|
7.2 | Ki | 25 | — | |
NDBJFFCSTXBTFV
|
7.2 | IC50 | 6 | — | |
NHFDRBXTEDBWCZ
|
7.2 | Ki | 41 | — | |
OSDSLNBKGDENNX
|
7.2 | IC50 | 3 | — | |
SACRIVBWIXWZAH
|
7.2 | Ki | 4 | — | |
XPPLYAKZGXYPOZ
|
7.2 | Ki | 6 | — | |
HVXKQKFEHMGHSL
|
7.2 | Kd | 21 | — | |
NIFOBCJOHDKDIO
|
7.2 | IC50 | 3 | — | |
APPXQUDJLJXULP
|
7.2 | IC50 | 47 | — | |
QOMGQLZYIUPQLG
|
7.2 | IC50 | 7 | — | |
WFJQCQNBWDAYSK
|
7.2 | IC50 | 4 | — | |
XPEVSMSGIHLOSK
|
7.2 | IC50 | 3 | — | |
QTBWCSQGBMPECM
|
7.2 | Kd | 21 | Yes |