Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CNTCGRJDUJEUDG
|
7.6 | Ki | 37 | — | |
CPHGZDSYMREPNQ
|
7.6 | IC50 | 6 | — | |
FLEAYYMORDPWAJ
|
7.6 | Ki | 90 | — | |
LGHBDVLAHHANMX
|
7.6 | Ki | 53 | — | |
MFMXAWQGPQXDRJ
|
7.6 | Ki | 27 | — | |
NKEUPUJTVALZIK
|
7.6 | Ki | 28 | — | |
RKGQENOGQBXEPA
|
7.6 | IC50 | 6 | — | |
VKQPTVJDZIILPG
|
7.6 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
7.6 | IC50 | 8 | Yes | |
ZAARMHXLYCHRAK
|
7.6 | Ki | 20 | — | |
DPMQHTABGLRCQK
|
7.6 | IC50 | 5 | — | |
PHXJVRSECIGDHY
|
7.6 | IC50 | 59 | — | |
GCIKSSRWRFVXBI
|
7.6 | Kd | 109 | Yes | |
AILRADAXUVEEIR
|
7.6 | IC50 | 75 | — | |
CTSDMCNSBRVZGJ
|
7.5 | IC50 | 7 | — | |
DKZYXHCYPUVGAF
|
7.5 | Kd | 112 | — | |
AICWWSFUNVNYGQ
|
7.5 | IC50 | 2 | — | |
VRQMAABPASPXMW
|
7.5 | Kd | 10 | — | |
FNHKPVJBJVTLMP
|
7.5 | IC50 | 29 | — | |
JNLSTLQFDDAULK
|
7.5 | IC50 | 4 | — | |
MLLQJNIKDWEEFT
|
7.5 | IC50 | 6 | — | |
ZVVQDNWRXSSQDL
|
7.5 | IC50 | 3 | — | |
BYSACNLCTNNHPN
|
7.5 | IC50 | 2 | — | |
NRBCZVLKKQZZNF
|
7.5 | IC50 | 2 | — | |
SKDBXDGKLQALIZ
|
7.5 | IC50 | 15 | — | |
UDFDIIVNIYWXDM
|
7.5 | Ki | 74 | — | |
VSVWQTDDGQSGHP
|
7.5 | Ki | 51 | — | |
WUWDLXZGHZSWQZ
|
7.5 | Ki | 41 | — | |
XMGFTZYNTYNOOJ
|
7.5 | Ki | 10 | — | |
YEHCNYAQEBQCCS
|
7.5 | Ki | 74 | — | |
ZCCJKVBTHCOISJ
|
7.5 | Ki | 46 | — | |
CSGQVNMSRKWUSH
|
7.5 | Kd | 21 | — | |
JCFYYOOCRKTOGG
|
7.5 | IC50 | 3 | — | |
UHTHHESEBZOYNR
|
7.5 | IC50 | 66 | Yes | |
YOHLRCOPRAVUCJ
|
7.5 | IC50 | 6 | — | |
COFRCLHJWNUSGM
|
7.4 | IC50 | 2 | — | |
UHKNINGWQKGQGB
|
7.4 | IC50 | 3 | — | |
XEDLQHAQDJOFQI
|
7.4 | IC50 | 2 | — | |
XYFPWWZEPKGCCK
|
7.4 | IC50 | 34 | — | |
IKZPPFXCBWIVPC
|
7.4 | IC50 | 3 | — | |
LBVKEEFIPBQIMD
|
7.4 | Ki | 27 | — | |
MFAQYJIYDMLAIM
|
7.4 | Kd | 130 | Yes | |
NXSJMRCTGYTSTK
|
7.4 | Kd | 200 | — | |
QKPLUKMJEKRAJD
|
7.4 | Ki | 30 | Yes | |
RTYJMUXLFRYRBU
|
7.4 | Ki | 35 | — | |
SYBRDWADIVSRRM
|
7.4 | IC50 | 2 | — | |
BNDYIYYKEIXHNK
|
7.4 | IC50 | 7 | Yes | |
PAFIGBIGZBXCGJ
|
7.4 | IC50 | 2 | — | |
YFVCYTODGMGPAD
|
7.4 | IC50 | 4 | — | |
ONIQOQHATWINJY
|
7.3 | IC50 | 25 | — |