Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXWNRDQAMADNES
|
7.8 | IC50 | 3 | — | |
QDIPGXPRBSWHHQ
|
7.8 | IC50 | 2 | — | |
TXFSECOZKAKHMC
|
7.8 | IC50 | 3 | — | |
UYXYKLOTLJDLNL
|
7.8 | IC50 | 4 | — | |
XIIOFHFUYBLOLW
|
7.8 | IC50 | 2 | — | |
XLSPYLMTRXPYKY
|
7.8 | IC50 | 13 | — | |
VSVJBCKLXDHEJV
|
7.8 | IC50 | 6 | — | |
GJKVMXDBPDDFHI
|
7.8 | Ki | 27 | — | |
GWMATETWMAQOFL
|
7.8 | Ki | 36 | — | |
PUPCRRRSBUYJAD
|
7.8 | Ki | 44 | Yes | |
TWZVBMXTDSNZLS
|
7.8 | Ki | 7 | — | |
RYYNGWLOYLRZLK
|
7.8 | Kd | 45 | — | |
NSZXLMVQBNISCL
|
7.8 | IC50 | 2 | — | |
XZXHXSATPCNXJR
|
7.8 | Kd | 165 | Yes | |
DZFZXPPHBWCXPQ
|
7.8 | IC50 | 12 | — | |
KVGTWUGUDPNRGC
|
7.7 | IC50 | 6 | — | |
NSKYYUZMAXEZIR
|
7.7 | Ki | 15 | — | |
RAKDOBWGYQVOPT
|
7.7 | IC50 | 2 | — | |
SQZDJBNTERGDSI
|
7.7 | IC50 | 5 | — | |
HIHOEGPXVVKJPP
|
7.7 | IC50 | 10 | — | |
HXHAJRMTJXHJJZ
|
7.7 | IC50 | 52 | Yes | |
MJHOMTRKVMKCNE
|
7.7 | IC50 | 12 | — | |
WINHZLLDWRZWRT
|
7.7 | Kd | 201 | Yes | |
BYSPSKYBWHPEJW
|
7.7 | IC50 | 6 | — | |
IXLOPQOCFOQEQN
|
7.7 | Ki | 2 | — | |
JSDGKSMNPHJDFK
|
7.7 | Ki | 35 | — | |
JZLUCFJMWJDRIK
|
7.7 | IC50 | 7 | — | |
KJRVCMVPIKELBC
|
7.7 | IC50 | 12 | — | |
MULNSLQVKKUPJN
|
7.7 | Ki | 41 | — | |
NFMGZVPRGVERNN
|
7.7 | Ki | 44 | — | |
NWKUBTQEYKTRNT
|
7.7 | IC50 | 4 | — | |
RAHBGWKEPAQNFF
|
7.7 | Kd | 26 | — | |
VCSQVKQFGYRGEH
|
7.7 | Ki | 13 | — | |
XKZQZMSAWVDRSP
|
7.7 | Ki | 39 | Yes | |
XNEPVLVYFUGJLF
|
7.7 | Ki | 27 | — | |
XYXLUJQBBIBJFV
|
7.7 | Ki | 36 | — | |
XIHXBNRAWIZORJ
|
7.7 | IC50 | 2 | — | |
FFPFOCJSSHPGFQ
|
7.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.7 | Kd | 213 | — | |
XTUBKDJMCMOXFL
|
7.7 | IC50 | 2 | — | |
HVKJROZQSCMKQH
|
7.7 | IC50 | 2 | — | |
SKMYNDYPMNSWDD
|
7.7 | IC50 | 2 | — | |
FJTQBVRKZLEDPK
|
7.7 | IC50 | 4 | — | |
FASQTICQHQVOKY
|
7.6 | IC50 | 3 | — | |
GUUYUIDTJAWAHO
|
7.6 | IC50 | 4 | — | |
IAYGCINLNONXHY
|
7.6 | Kd | 50 | — | |
VVXPVDHTIYRFQN
|
7.6 | IC50 | 2 | — | |
CTNPALGJUAXMMC
|
7.6 | Kd | 151 | — | |
JIBBGYSUSKAPDY
|
7.6 | IC50 | 19 | — | |
MHITTXFPZXWLMH
|
7.6 | Kd | 6 | — |