Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SVRNPAWUQSRQDR
|
8.1 | IC50 | 2 | — | |
JCCUAVDBGXASEC
|
8.1 | IC50 | 3 | — | |
BHDNMZNYEGULRO
|
8.1 | IC50 | 2 | — | |
ALKJNCZNEOTEMP
|
8.1 | Kd | 55 | — | |
OIIPLUSQGIIGMV
|
8.1 | IC50 | 2 | — | |
WOSKHXYHFSIKNG
|
8.1 | IC50 | 24 | — | |
YLJPQGVBJWZONC
|
8.1 | IC50 | 6 | — | |
HHXNFVOVAOZPLV
|
8.0 | IC50 | 3 | — | |
ZBZATSVLKXDTMV
|
8.0 | IC50 | 3 | — | |
BLQYVHBZHAISJM
|
8.0 | IC50 | 54 | — | |
CVWXJKQAOSCOAB
|
8.0 | Kd | 35 | — | |
FTDWSWREBGYXDZ
|
8.0 | IC50 | 10 | — | |
NRGYZNJPCGRCLV
|
8.0 | Ki | 52 | — | |
PTVPBWWDGZSEAF
|
8.0 | Ki | 63 | — | |
RWEHAHIEUDLKGT
|
8.0 | Ki | 33 | — | |
SBLMCLDRWJNEJK
|
8.0 | IC50 | 17 | — | |
SRUYMJRFVGLQDV
|
8.0 | Ki | 37 | — | |
WPXVVAWAHQHJPF
|
8.0 | IC50 | 41 | — | |
WYCSRUVPJUYDGP
|
8.0 | IC50 | 6 | — | |
YFNWWNRZJGMDBR
|
8.0 | Kd | 35 | — | |
ZGDSBEUMPIMXBM
|
8.0 | Ki | 42 | — | |
ZKHDDJKHTPLPOQ
|
8.0 | Ki | 62 | — | |
ZXLFIHLBHMLHFJ
|
8.0 | Ki | 31 | — | |
SZTLWJSWANAPBP
|
8.0 | IC50 | 2 | — | |
VWCZORWQNKCYGE
|
8.0 | IC50 | 17 | — | |
SZFYZDIPRMLBDC
|
8.0 | IC50 | 9 | — | |
QJOKMKBZEMLHIM
|
8.0 | IC50 | 5 | — | |
XACVMSVOYKULCV
|
8.0 | IC50 | 2 | — | |
NTUNMKNXRUDCPX
|
8.0 | IC50 | 2 | — | |
ZVPDNRVYHLRXLX
|
8.0 | IC50 | 35 | Yes | |
QCOUFOILFGCFOO
|
8.0 | IC50 | 2 | — | |
VYZPFLWPKPMFKB
|
8.0 | IC50 | 2 | — | |
ZUSOUYHYDDCGIC
|
8.0 | IC50 | 4 | — | |
IKMBEAVQWGZKRA
|
7.9 | IC50 | 2 | — | |
QCHOFSGKMWUAPT
|
7.9 | IC50 | 2 | — | |
IDGNCVHQDDOPND
|
7.9 | IC50 | 6 | — | |
SPMVMDHWKHCIDT
|
7.9 | Kd | 30 | — | |
BOBGABAXWFYHQX
|
7.9 | Ki | 9 | — | |
GCYXEGSPUDSZJY
|
7.9 | Ki | 82 | — | |
JTRNNNVASYCTLO
|
7.9 | Ki | 14 | — | |
MVJMMLFMPWITEJ
|
7.9 | Ki | 110 | — | |
UOVCGJXDGOGOCZ
|
7.9 | Ki | 59 | — | |
MLDQJTXFUGDVEO
|
7.9 | IC50 | 85 | Yes | |
WGBQSNXDFBWRGI
|
7.9 | IC50 | 2 | — | |
BNPMMVDYMYENIM
|
7.9 | IC50 | 4 | — | |
MKONGHOXTWPRPY
|
7.9 | IC50 | 2 | — | |
GVIULWWJXLMODX
|
7.9 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.9 | IC50 | 64 | Yes | |
XXEMOIBQTAXQNA
|
7.9 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
7.8 | Kd | 289 | Yes |