Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WQTDKOSNNMUDQK
|
8.3 | IC50 | 5 | — | |
XJSFDMGICAWQFS
|
8.3 | Ki | 60 | — | |
ZZLHNPULFZMEMI
|
8.3 | IC50 | 2 | — | |
BLYRPGBSIKAIAU
|
8.3 | IC50 | 24 | Yes | |
OKQBSSHHQHTUOB
|
8.3 | IC50 | 2 | — | |
YXARVHZXTQVAOP
|
8.3 | IC50 | 11 | — | |
CRQNIBKIWTWDFL
|
8.3 | IC50 | 3 | — | |
HXOYQIBZUSAYOZ
|
8.2 | IC50 | 2 | — | |
SQXGUVZOXXNPJG
|
8.2 | IC50 | 2 | — | |
VTWWRKFUHCSCEW
|
8.2 | Kd | 19 | — | |
XHXOJKOXEKXDSQ
|
8.2 | IC50 | 5 | Yes | |
ACNNJWMMLBYERQ
|
8.2 | IC50 | 2 | — | |
GNMDVOZMYIYNJR
|
8.2 | IC50 | 2 | — | |
AKWLDQDWZNJYKL
|
8.2 | IC50 | 14 | — | |
AVQNZSIEXOYAGE
|
8.2 | IC50 | 6 | — | |
FOLXFWBVNHRGIV
|
8.2 | IC50 | 6 | — | |
SHAHCUNTVXETOK
|
8.2 | IC50 | 2 | — | |
UKYJKXMPIDEQFF
|
8.2 | IC50 | 16 | — | |
XQYRIHGWAJPTNC
|
8.2 | IC50 | 2 | — | |
WOEVJDXDZJWENO
|
8.2 | IC50 | 3 | — | |
ZLLYPULBPHUOLR
|
8.2 | IC50 | 2 | — | |
SHDOSPHGKDEPQN
|
8.2 | IC50 | 2 | — | |
UNQRFBPIZOYNKG
|
8.2 | IC50 | 2 | — | |
KDGFLJKFZUIJMX
|
8.2 | IC50 | 10 | — | |
JONUUBFCZUAOFY
|
8.2 | IC50 | 10 | — | |
WPHKIQPVPYJNAX
|
8.2 | IC50 | 81 | — | |
PBMFNTXIZOOABV
|
8.1 | IC50 | 2 | — | |
UDYNQUNBJNMHEA
|
8.1 | IC50 | 2 | — | |
YRUDYNCGPZHXRB
|
8.1 | Kd | 6 | — | |
YOBIWCLAYQWPPW
|
8.1 | IC50 | 23 | — | |
FGFZBTQWDLZHSI
|
8.1 | IC50 | 4 | — | |
MHZIGJBWNNGGBZ
|
8.1 | IC50 | 3 | — | |
RNIXZCQWBPDHPR
|
8.1 | IC50 | 3 | — | |
VVEWWOOATHIBFT
|
8.1 | IC50 | 2 | — | |
XXJWYDDUDKYVKI
|
8.1 | Kd | 52 | — | |
LVLFSSZNAIKYCD
|
8.1 | IC50 | 19 | — | |
BETBNWGUKZUUAX
|
8.1 | IC50 | 21 | — | |
BHSOPYVVEZFHDB
|
8.1 | Ki | 25 | Yes | |
DZSUJUOJJJCWGG
|
8.1 | Ki | 55 | Yes | |
FDVSOQRNTAPCHB
|
8.1 | Ki | 40 | — | |
HLOASMXRJBZZAG
|
8.1 | IC50 | 3 | — | |
IFPPYSWJNWHOLQ
|
8.1 | Ki | 52 | Yes | |
NECQZMQPXFYVOY
|
8.1 | Ki | 26 | — | |
NOAXCXNLWPVHFH
|
8.1 | IC50 | 2 | — | |
PROLIXHVRCJEFH
|
8.1 | Ki | 46 | — | |
QXIOZIFTPMAING
|
8.1 | IC50 | 17 | — | |
SDBOIBYRBWPIEL
|
8.1 | Ki | 31 | — | |
TVUWQDLBEOZVOU
|
8.1 | Ki | 41 | — | |
WFTZMAAMCVPJJT
|
8.1 | Ki | 26 | — | |
CIDPAEWKWWPDKH
|
8.1 | IC50 | 2 | — |