Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MWKSRKSEWLRPBL
|
8.6 | Kd | 1075 | — | |
BLMSWRQOCWCQDM
|
8.5 | IC50 | 2 | — | |
BVHZLDLRNBQWRF
|
8.5 | IC50 | 5 | — | |
KXMZDGSRSGHMMK
|
8.5 | IC50 | 14 | — | |
OEUMLQMTMOCCGW
|
8.5 | Kd | 6 | — | |
VWDJZFSVNMUGSS
|
8.5 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
8.5 | Ki | 44 | — | |
CXBBWVXSZINRCS
|
8.5 | Ki | 41 | — | |
NIKNJFKATRPZSL
|
8.5 | Ki | 9 | — | |
OWFXKTOLFUQPDJ
|
8.5 | Ki | 36 | — | |
RBXYGQNZRVPDNB
|
8.5 | Ki | 34 | — | |
RYYNGWLOYLRZLK
|
8.5 | Ki | 104 | — | |
VCZWRJVZJHBRFC
|
8.5 | IC50 | 2 | — | |
XKZINYYXWJEYEL
|
8.5 | Ki | 37 | — | |
ZWVZORIKUNOTCS
|
8.5 | Ki | 69 | — | |
FIDOSJXSMFKBQH
|
8.5 | IC50 | 2 | — | |
IUCMEDMSUCVZQN
|
8.5 | IC50 | 2 | — | |
LOLPPWBBNUVNQZ
|
8.5 | IC50 | 97 | Yes | |
ZTIHSLVMCONHQU
|
8.5 | IC50 | 5 | — | |
QGWFBTCMBJQAGH
|
8.5 | IC50 | 2 | — | |
LRJJEMRURFIKDD
|
8.4 | IC50 | 6 | — | |
FWEAPVSZAHZTHG
|
8.4 | IC50 | 2 | — | |
BMTDMPCSMBKKPW
|
8.4 | Kd | 2 | — | |
KVXVWTTVVQJNLT
|
8.4 | IC50 | 2 | — | |
FFCFHBVSGILIJY
|
8.4 | Ki | 17 | — | |
NWAUBAGBGOPJLF
|
8.4 | Ki | 51 | Yes | |
OFUBWOTWQPAEDG
|
8.4 | IC50 | 6 | — | |
OFXSDEOZNJESCC
|
8.4 | IC50 | 2 | — | |
OUDNHJQPMQFCDI
|
8.4 | IC50 | 4 | — | |
OWRXHGAFWZFFCW
|
8.4 | Ki | 113 | — | |
UEJXELMBDCXXAQ
|
8.4 | IC50 | 9 | — | |
XOOAAYRIVATZNM
|
8.4 | Ki | 55 | — | |
YHVHYWYQEFELOW
|
8.4 | IC50 | 44 | — | |
KHAIGKZESPRVDY
|
8.4 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
8.4 | Kd | 220 | — | |
BSQGOBUXBCHTJR
|
8.4 | IC50 | 2 | — | |
DKNUPRMJNUQNHR
|
8.4 | IC50 | 33 | — | |
GAQUZKVNFLINTC
|
8.4 | IC50 | 2 | — | |
QLRRJMOBVVGXEJ
|
8.4 | IC50 | 2 | — | |
ULNQWYGVWVDLPK
|
8.4 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
8.3 | Kd | 153 | — | |
FHZCSNTVCRCIKT
|
8.3 | IC50 | 3 | — | |
MVQAYSXDCGCOIE
|
8.3 | IC50 | 2 | — | |
BGVQPQHIUOTLBT
|
8.3 | Kd | 6 | — | |
GPXBXXGIAQBQNI
|
8.3 | IC50 | 11 | — | |
XYJGSYPUEAFKLG
|
8.3 | IC50 | 2 | — | |
CUDVHEFYRIWYQD
|
8.3 | Kd | 11 | — | |
NGOUBNKIABYCRY
|
8.3 | IC50 | 2 | — | |
NWMPVMMGSHXANZ
|
8.3 | Ki | 58 | — | |
QRUAIHIOEIIASP
|
8.3 | IC50 | 2 | — |