Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEJGTFPOEJWEGG
|
9.0 | Kd | 149 | — | |
DYLOIFYWXMEMOK
|
8.9 | IC50 | 2 | — | |
KMHRABISHFQKDA
|
8.9 | IC50 | 2 | — | |
LBELDIIRDVZLHQ
|
8.9 | IC50 | 2 | — | |
WMWHVTDZNIVNIE
|
8.9 | IC50 | 9 | — | |
WMWHVTDZNIVNIE
|
8.9 | IC50 | 9 | — | |
LMFNJXLDISVWLF
|
8.9 | IC50 | 5 | — | |
NVRXTLZYXZNATH
|
8.9 | Ki | 47 | Yes | |
DIMALNWQSQDLJJ
|
8.9 | IC50 | 3 | — | |
MPYUMMWCLQVMLG
|
8.9 | IC50 | 11 | — | |
BJGZYOBYHRNCMW
|
8.8 | IC50 | 2 | — | |
PCOBMDHMIYSEJY
|
8.8 | IC50 | 2 | — | |
XFPDCDUJYXKATF
|
8.8 | IC50 | 2 | — | |
ADFZKKWKESWUFY
|
8.8 | IC50 | 8 | — | |
BEXCPFCIYIOGDW
|
8.8 | IC50 | 2 | — | |
OMWMITRWODCQFK
|
8.8 | IC50 | 3 | — | |
VIVXZYGJUYINGG
|
8.8 | IC50 | 2 | — | |
CXQHYVUVSFXTMY
|
8.8 | Kd | 154 | — | |
DZUFTTMDQLYMBE
|
8.8 | IC50 | 10 | Yes | |
KUNZDWIFPOMUOX
|
8.8 | Ki | 36 | — | |
VKBFHTIUXUCYRQ
|
8.8 | Ki | 66 | — | |
XKFTZKGMDDZMJI
|
8.8 | Ki | 56 | — | |
LRICQCBDYKWUDI
|
8.8 | IC50 | 2 | — | |
ITONFAYEXGFEEK
|
8.8 | IC50 | 2 | — | |
YRBWLEAMGAGYBK
|
8.8 | IC50 | 6 | — | |
MANWCWXDWLXTDJ
|
8.7 | IC50 | 2 | — | |
OBWIGYYOZSWZCZ
|
8.7 | IC50 | 2 | — | |
PCNMRGUJZFWHPU
|
8.7 | IC50 | 2 | — | |
XIWHTFJGIGNJFL
|
8.7 | IC50 | 2 | — | |
FTUPHXIFYRNJMA
|
8.7 | IC50 | 2 | — | |
AMHUBFWCCMLLCJ
|
8.7 | IC50 | 15 | — | |
NAHKSTDKHZOXFT
|
8.7 | IC50 | 2 | — | |
YYYBQWITTVLVFM
|
8.7 | IC50 | 2 | — | |
GQOCBCGJBHCFFD
|
8.7 | IC50 | 2 | — | |
IDXKJSSOUXWLDB
|
8.7 | IC50 | 2 | — | |
RKGOHOXKHIGYOL
|
8.7 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 118 | — | |
RQJGLDQSQBZHDJ
|
8.6 | IC50 | 2 | — | |
BDHJKYLJPYEWOX
|
8.6 | IC50 | 2 | — | |
XPYLIJSVMCGXKI
|
8.6 | IC50 | 2 | — | |
CTRGHKNEFBXHLG
|
8.6 | IC50 | 2 | — | |
DKSNLQYRZJKYOC
|
8.6 | Ki | 51 | — | |
KGSRYTUWXUESJK
|
8.6 | IC50 | 7 | — | |
OSZVHJYNXBUVAH
|
8.6 | IC50 | 12 | — | |
WINHZLLDWRZWRT
|
8.6 | Ki | 66 | — | |
FVYFIPZMFFIGOO
|
8.6 | IC50 | 2 | — | |
IIEOPFUEUQSIJW
|
8.6 | IC50 | 2 | — | |
RGECMCDLOXPBCC
|
8.6 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
8.6 | IC50 | 408 | — | |
GUBJNPWVIUFSTR
|
8.6 | Kd | 103 | — |