Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YLQMVIRZBOJBCV
|
6.2 | IC50 | 7 | Yes | |
XISIJMIPHPQCQQ
|
6.2 | IC50 | 9 | — | |
AYCPARAPKDAOEN
|
6.1 | Kd | 73 | — | |
HOZUXBLMYUPGPZ
|
6.1 | IC50 | 3 | Yes | |
OONFNUWBHFSNBT
|
6.1 | IC50 | 11 | — | |
UORAPQCBWYIISR
|
6.1 | IC50 | 12 | — | |
BEMNJULZEQTDJY
|
6.1 | Kd | 8 | — | |
LOGJQOUIVKBFGH
|
6.1 | IC50 | 11 | Yes | |
BKBCSMDCCAWWNC
|
6.1 | Ki | 7 | — | |
CHTMRWQLNNRRFJ
|
6.1 | Ki | 70 | — | |
DJRPFIWIDKXORZ
|
6.1 | Ki | 9 | — | |
HHSVICUMCOBRPT
|
6.1 | Ki | 33 | — | |
IFQICUARAXVEIQ
|
6.1 | Ki | 18 | — | |
IUEBPIPDFMCSTP
|
6.1 | Ki | 29 | — | |
JCZBWICLNFNCMR
|
6.1 | Ki | 9 | — | |
JHYHWHUTTXJICB
|
6.1 | Ki | 18 | — | |
JRLSUZIPUYDUKX
|
6.1 | Ki | 22 | — | |
NLUPJKQOKWBWFC
|
6.1 | Ki | 69 | — | |
VRIFJAKXSBXYFZ
|
6.1 | Ki | 8 | — | |
XKXPQPXJZUDSOG
|
6.1 | IC50 | 2 | — | |
XSRHBCYNCKAFKS
|
6.1 | Ki | 45 | — | |
YACXOXQTGJXYNX
|
6.1 | Ki | 11 | — | |
DYNHJHQFHQTFTP
|
6.1 | Kd | 38 | — | |
OMZCMEYTWSXEPZ
|
6.1 | Kd | 43 | Yes | |
HHZIURLSWUIHRB
|
6.1 | Kd | 57 | Yes | |
CXISENKPXGMZEE
|
6.0 | IC50 | 4 | — | |
SHPFDGWALWEPGS
|
6.0 | Kd | 35 | — | |
BCTIPSBBPQBXAG
|
6.0 | IC50 | 4 | — | |
VBYMFAOTZHNONG
|
6.0 | IC50 | 5 | — | |
XUZMWHLSFXCVMG
|
6.0 | Kd | 24 | — | |
AGSASGLZNILGCY
|
6.0 | Ki | 3 | — | |
AHZUHDSHQGQZRW
|
6.0 | IC50 | 4 | Yes | |
DLWMVUDMPMKGEE
|
6.0 | Ki | 24 | — | |
FXXMEMJTLOATRB
|
6.0 | Ki | 5 | — | |
HAIHTRCFSLFERU
|
6.0 | IC50 | 3 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
IZFIXANBEYSEOB
|
6.0 | IC50 | 5 | — | |
JWQXXOLUOCHGFG
|
6.0 | IC50 | 5 | — | |
KDKUVYLMPJIGKA
|
6.0 | Kd | 91 | Yes | |
KTEIFNKAUNYNJU
|
6.0 | Ki | 48 | — | |
KTQYQHLIMZOBSM
|
6.0 | Ki | 12 | — | |
LDHYCINFJPCBRY
|
6.0 | Ki | 9 | — | |
MHRZYVYAAMLZJC
|
6.0 | Ki | 4 | — | |
NJPWCTYVEJIQBM
|
6.0 | Ki | 72 | — | |
NMHMCXTYPRADBA
|
6.0 | Ki | 20 | — | |
OPLHMHMCXQXEQG
|
6.0 | Ki | 10 | — | |
PPCNMZPSQZFFGM
|
6.0 | Ki | 8 | — | |
TUDIKYFSCUIAIT
|
6.0 | Ki | 8 | — | |
UQABTPYYEALKPO
|
6.0 | IC50 | 2 | Yes | |
VJKJKZOWXJKSSK
|
6.0 | Ki | 4 | — |