Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DZGATJHVQUFYSK
|
6.4 | Ki | 12 | — | |
GEGCXGMFUYJULA
|
6.4 | Ki | 30 | Yes | |
HZPACYSNLOCDLW
|
6.4 | Ki | 48 | — | |
JCFJQIHDZHHMQT
|
6.4 | Ki | 42 | — | |
KUCNBQPAJZRQMJ
|
6.4 | IC50 | 11 | — | |
SRROIPFGGDHJCJ
|
6.4 | Ki | 7 | — | |
UYJNQQDJUOUFQJ
|
6.4 | Ki | 68 | — | |
VERWOWGGCGHDQE
|
6.4 | IC50 | 23 | — | |
WUBHCQHBUVGGRX
|
6.4 | Ki | 11 | — | |
ZBYGBITZFKOQTA
|
6.4 | Ki | 18 | — | |
ZLHFILGSQDJULK
|
6.4 | Ki | 37 | Yes | |
ISABFXAQXIFBSS
|
6.4 | IC50 | 3 | — | |
OTTCBLPTHPBEEX
|
6.4 | Ki | 11 | Yes | |
HFNKQEVNSGCOJV
|
6.4 | Kd | 65 | — | |
ZZOIXVRJVONVLW
|
6.4 | IC50 | 4 | — | |
CXNXNSYZZDJASK
|
6.4 | IC50 | 4 | — | |
HFNKQEVNSGCOJV
|
6.3 | Ki | 18 | — | |
SEZFNTZQMWJIAI
|
6.3 | IC50 | 9 | Yes | |
ZYTRQJFBKVMEAK
|
6.3 | IC50 | 2 | — | |
AYXVSCVVQIADBF
|
6.3 | Ki | 10 | — | |
IFWNPAWLKUVJGK
|
6.3 | IC50 | 3 | — | |
LUPCHAFIKZSOOK
|
6.3 | Ki | 15 | — | |
NOBMKUVHFRVBES
|
6.3 | Ki | 19 | — | |
UGUZOLHBLLTLBA
|
6.3 | Ki | 15 | — | |
YEPNVBNYCRGZRX
|
6.3 | Ki | 26 | — | |
ZLVOTRRGLSDLPF
|
6.3 | Ki | 36 | — | |
PBCZSGKMGDDXIJ
|
6.3 | Kd | 68 | Yes | |
VDXGLZJPQRGNLY
|
6.3 | IC50 | 10 | — | |
MJQGHLODJHABRA
|
6.3 | IC50 | 10 | — | |
OYONTEXKYJZFHA
|
6.3 | Kd | 69 | Yes | |
ZBNZXTGUTAYRHI
|
6.3 | Kd | 102 | Yes | |
VNBRGSXVFBYQNN
|
6.2 | IC50 | 22 | Yes | |
PABMYTICQCKZAG
|
6.2 | IC50 | 3 | — | |
QBRQTJMZEYORSP
|
6.2 | Kd | 12 | — | |
USPKFTCYXHJXCN
|
6.2 | IC50 | 4 | — | |
NWXGFDVFXJMUDD
|
6.2 | IC50 | 5 | — | |
ULTCRVJUAZCGPP
|
6.2 | IC50 | 5 | — | |
CQFVDHNTTRWVQD
|
6.2 | Ki | 9 | — | |
ILUGAYBMBIJXHC
|
6.2 | Ki | 9 | — | |
LJKJYKWDLJUZHA
|
6.2 | Ki | 24 | — | |
QCOULMVHIHJKFY
|
6.2 | Ki | 14 | — | |
QRWHFUYBHXDYNV
|
6.2 | Ki | 2 | — | |
RPGBQFNDFPEOON
|
6.2 | Ki | 22 | — | |
STUPRWVTVIXNLF
|
6.2 | Ki | 6 | — | |
VWACUNWBMWWMPJ
|
6.2 | Ki | 18 | — | |
JGEBLDKNWBUGRZ
|
6.2 | IC50 | 20 | Yes | |
RMTJSBZCZKCYHB
|
6.2 | IC50 | 13 | — | |
KOZFSFOOLUUIGY
|
6.2 | Kd | 88 | Yes | |
LQVXSNNAFNGRAH
|
6.2 | Kd | 33 | Yes | |
TXSZGBMOPCXBTP
|
6.2 | IC50 | 7 | Yes |