Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MAGVRNDWTTZRHB
|
6.7 | IC50 | 2 | — | |
OPRQSQDMYPVYOV
|
6.7 | IC50 | 7 | — | |
NWCCWSWQAFETLG
|
6.7 | IC50 | 4 | — | |
SEZFNTZQMWJIAI
|
6.7 | Ki | 22 | — | |
FLBNLJLONKAPLR
|
6.6 | Kd | 31 | — | |
DZPXNXYARLTMGL
|
6.6 | IC50 | 2 | — | |
MVCOAUNKQVWQHZ
|
6.6 | Kd | 54 | Yes | |
PDOQBOJDRPLBQU
|
6.6 | Kd | 21 | — | |
VVYFYJMXONNWBA
|
6.6 | IC50 | 7 | Yes | |
ZZSBPGIGIUFJRA
|
6.6 | Kd | 46 | — | |
CACMTVGXYAZZNY
|
6.6 | Ki | 11 | — | |
CKVWQORGCCEYHS
|
6.6 | Ki | 50 | — | |
RIUZPIBUSOHUKF
|
6.6 | Ki | 23 | — | |
WVFWTUJEHMVUBG
|
6.6 | Ki | 25 | — | |
XPHWIERLJBFPFV
|
6.6 | Ki | 69 | — | |
XZWVOUQIYLZUCJ
|
6.6 | Ki | 23 | — | |
DUKJABPGWUISRC
|
6.6 | IC50 | 10 | — | |
CUIHSIWYWATEQL
|
6.6 | Kd | 61 | Yes | |
GADRFNSBFFQCNB
|
6.6 | IC50 | 2 | — | |
OQBJXGADOAMRSR
|
6.5 | IC50 | 5 | — | |
XYONNOXYJMPBMA
|
6.5 | IC50 | 2 | — | |
AUDNGNGLLRZLDR
|
6.5 | Ki | 33 | — | |
BPJQSSSZFGZEOF
|
6.5 | Ki | 4 | — | |
FMPKTXNCNJCHCC
|
6.5 | Ki | 25 | — | |
FXQWJULRETZHHW
|
6.5 | Ki | 14 | — | |
GQGMUKOYILWOIQ
|
6.5 | Ki | 25 | — | |
GXJSLIOOPZRPEV
|
6.5 | Ki | 34 | — | |
JISZKDFLHFISOW
|
6.5 | Ki | 6 | — | |
JJGSOVIZOMZMCS
|
6.5 | Ki | 35 | — | |
JNXJKTXDSPWNRP
|
6.5 | Ki | 30 | — | |
KJVWCDAPVMWKLJ
|
6.5 | Ki | 20 | — | |
LXVBELDBJGYFEM
|
6.5 | Ki | 20 | — | |
MZDKLVOWGIOKTN
|
6.5 | Ki | 80 | — | |
NHFDRBXTEDBWCZ
|
6.5 | Kd | 12 | Yes | |
PKCDDUHJAFVJJB
|
6.5 | Ki | 13 | — | |
TVLFEDKEAOXRCZ
|
6.5 | Ki | 22 | — | |
UIRCQOKSJDLYBB
|
6.5 | Ki | 50 | — | |
VIJBEUTVNBPGIU
|
6.5 | Ki | 19 | — | |
ZGDYBJXDIXVTLV
|
6.5 | Ki | 54 | — | |
AAKJLRGGTJKAMG
|
6.5 | Kd | 50 | Yes | |
DJYWRQSMWCFDQX
|
6.5 | IC50 | 3 | — | |
SCMJNQHUUQLKRS
|
6.5 | IC50 | 5 | — | |
IWDBZVDOUJFIND
|
6.5 | IC50 | 5 | — | |
WCWUXEGQKLTGDX
|
6.4 | Kd | 22 | Yes | |
IGRYEDIMNMEBBU
|
6.4 | IC50 | 9 | — | |
DFJSJLGUIXFDJP
|
6.4 | Kd | 9 | — | |
FGTCROZDHDSNIO
|
6.4 | Kd | 5 | — | |
FHFKMBKXODPUFW
|
6.4 | IC50 | 5 | — | |
HAYYBYPASCDWEQ
|
6.4 | IC50 | 47 | — | |
LCVIRAZGMYMNNT
|
6.4 | Kd | 20 | — |