Target Details
| UniProt AC | P07949 |
|---|---|
| Gene Symbol | RET |
| Protein Name | Proto-oncogene tyrosine-protein kinase receptor Ret |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00028 (Cadherin) PF07714 (PK_Tyr_Ser-Thr) PF17756 (RET_CLD1) PF17812 (RET_CLD3) PF17813 (RET_CLD4) PF22540 (RET_CRD) |
Summary
- Multi-target molecules 656
- Clinical molecules 78
- Avg pChEMBL 7.52
KEGG Pathways (7)
Associated Diseases (6)
Active Molecules (656)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SOLRFWOVULTERW
|
6.9 | IC50 | 2 | — | |
DPAOHEUWPLGQDY
|
6.9 | IC50 | 4 | Yes | |
AEYLJTAIDDIOBA
|
6.9 | Ki | 53 | — | |
ATGVCJYHNOSZEV
|
6.9 | Ki | 23 | — | |
CJUJLGFTKBBDMG
|
6.9 | Ki | 9 | — | |
NCPXFACDZCEIQL
|
6.9 | Ki | 7 | — | |
PDBPUXLUVDSLML
|
6.9 | Ki | 14 | — | |
PYXQMJSGJIJHJT
|
6.9 | Ki | 28 | — | |
ZGZVRPRSFXRGCF
|
6.9 | Ki | 76 | — | |
AAQXIFQQTLXRNG
|
6.9 | IC50 | 2 | — | |
BMGQWWVMWDBQGC
|
6.9 | Kd | 147 | Yes | |
UJBJWYNPUOLFIZ
|
6.9 | IC50 | 49 | — | |
CJWIBINTCNTMJT
|
6.8 | IC50 | 4 | — | |
LTTAHJWMYYUXHI
|
6.8 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.8 | Kd | 231 | Yes | |
VBYCLUNCQJLFHE
|
6.8 | IC50 | 4 | Yes | |
BUMVKPFMQPYNEV
|
6.8 | IC50 | 3 | — | |
FQIRYXKZWMEKES
|
6.8 | IC50 | 8 | — | |
LYXOBSREVZDKST
|
6.8 | IC50 | 9 | — | |
AIQDZMUPVYDVLB
|
6.8 | Ki | 48 | — | |
GFFVAKKFWQHFLB
|
6.8 | IC50 | 5 | — | |
JCJSAFZMXVQVBR
|
6.8 | IC50 | 11 | Yes | |
RITAVMQDGBJQJZ
|
6.8 | Ki | 33 | — | |
SBFPHSVZEXSHTL
|
6.8 | Ki | 62 | — | |
WYOMXSAYYXBPMN
|
6.8 | Ki | 24 | — | |
BWXISLRRARTIGU
|
6.8 | IC50 | 6 | — | |
ZHMXXVNQAFCXKK
|
6.8 | IC50 | 15 | — | |
HAWQJVUHZAYNCF
|
6.8 | IC50 | 5 | — | |
WUWDLXZGHZSWQZ
|
6.8 | IC50 | 11 | Yes | |
UQRCJCNVNUFYDX
|
6.8 | Kd | 27 | — | |
OUKYUETWWIPKQR
|
6.8 | Kd | 31 | Yes | |
BJHCYTJNPVGSBZ
|
6.7 | IC50 | 5 | Yes | |
BPNUQXPIQBZCMR
|
6.7 | Kd | 83 | Yes | |
CMGWPZPIBTZFRI
|
6.7 | IC50 | 2 | — | |
GITWBPKQKQFIAW
|
6.7 | IC50 | 2 | — | |
GNRQZQLDSXCQET
|
6.7 | IC50 | 2 | — | |
CZQVOIDVDAVDFW
|
6.7 | Ki | 18 | — | |
DBXGGXLBTWZXBB
|
6.7 | Ki | 39 | — | |
GLDPXWNDIUPOHH
|
6.7 | IC50 | 6 | Yes | |
GQLWKGVBOIYMTN
|
6.7 | Ki | 35 | — | |
GXKYSFQMTTZPGW
|
6.7 | Ki | 7 | — | |
QBKUOOQFSVMDPB
|
6.7 | Ki | 31 | — | |
QLWUDWMYFSWGHK
|
6.7 | Ki | 22 | — | |
QNUKRWAIZMBVCU
|
6.7 | Ki | 46 | — | |
VNDWQCSOSCCWIP
|
6.7 | Ki | 39 | Yes | |
WQFGNANQTYLQBP
|
6.7 | Ki | 16 | — | |
XFWUTMHVDGPWLH
|
6.7 | Ki | 75 | — | |
XGMWRIIMIJPGBH
|
6.7 | Ki | 10 | — | |
BMGQWWVMWDBQGC
|
6.7 | Kd | 91 | Yes | |
BWCCBKUPFRNBAM
|
6.7 | IC50 | 2 | — |