Target Details
| UniProt AC | P07948 |
|---|---|
| Gene Symbol | LYN |
| Protein Name | Tyrosine-protein kinase Lyn |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 474
- Clinical molecules 117
- Avg pChEMBL 6.97
KEGG Pathways (13)
- B cell receptor signaling pathway
- Chemokine signaling pathway
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- IgSF CAM signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Long-term depression
- NF-kappa B signaling pathway
- Platelet activation
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JOOXLOJCABQBSG
|
6.3 | Kd | 139 | — | |
KOHNRDPXFDZZJF
|
6.3 | Ki | 31 | — | |
LRLDYTTWQIFWBD
|
6.3 | Ki | 25 | — | |
OLUKILHGKRVDCT
|
6.3 | Ki | 44 | Yes | |
PCQMERRARZKTPW
|
6.3 | Ki | 68 | — | |
QDOBTYVGPGFRCM
|
6.3 | Ki | 11 | — | |
UWDBNTXEKYRMSG
|
6.3 | Ki | 26 | — | |
WUWDLXZGHZSWQZ
|
6.3 | Ki | 41 | — | |
YDWMUCKJUNLURC
|
6.3 | Ki | 24 | — | |
YEPNVBNYCRGZRX
|
6.3 | Ki | 26 | — | |
ZGZVRPRSFXRGCF
|
6.3 | Ki | 76 | — | |
AAKJLRGGTJKAMG
|
6.3 | Kd | 50 | Yes | |
CSCOHEYTBLBQMG
|
6.3 | IC50 | 7 | Yes | |
TUKOILYAIRACKC
|
6.3 | IC50 | 7 | Yes | |
OJZKUAGKHXFNTK
|
6.3 | IC50 | 2 | — | |
RDFXBYJUHGEYHA
|
6.3 | IC50 | 9 | Yes | |
AHSDSYPFNQKAMQ
|
6.3 | IC50 | 2 | — | |
ANIANGUDIUAQEW
|
6.3 | IC50 | 2 | — | |
BDNQKKRHQCSPEM
|
6.3 | IC50 | 3 | — | |
BHHWCFSANVGEKE
|
6.3 | IC50 | 3 | — | |
BLIFHUIJBLJXIQ
|
6.3 | IC50 | 2 | — | |
BWHUGMDYLIIOLN
|
6.3 | IC50 | 2 | — | |
CQADGYMRJAVKJA
|
6.3 | IC50 | 2 | — | |
DKPXGWFFGXMEDV
|
6.3 | IC50 | 3 | — | |
DMBJCEFMXWJWAL
|
6.3 | IC50 | 2 | — | |
DPZGKYJHTOSMIA
|
6.3 | IC50 | 8 | — | |
FDVSTEYUPJGXHB
|
6.3 | IC50 | 2 | — | |
FNNHKBJKOSDELC
|
6.3 | IC50 | 2 | — | |
FPUDQJVLFVSZSC
|
6.3 | IC50 | 2 | — | |
GFQNQGIHFZEYTQ
|
6.3 | IC50 | 3 | — | |
HGDBRPWKZKQYJJ
|
6.3 | IC50 | 2 | — | |
HLHICHWQRZZBDS
|
6.3 | IC50 | 2 | — | |
HVZZKZIYGDQODO
|
6.3 | IC50 | 2 | — | |
JIHOLWSGBOJOLS
|
6.3 | IC50 | 3 | — | |
JNCYOWVWEITKGC
|
6.3 | IC50 | 2 | — | |
JRNKIJNZHPVJDT
|
6.3 | IC50 | 2 | — | |
KZRDVFBPXXGSPD
|
6.3 | IC50 | 9 | — | |
LJRBXGZFMWMQNY
|
6.3 | IC50 | 4 | — | |
LNHCWEMWGGTYRO
|
6.3 | IC50 | 3 | — | |
LPPUPUBHCBCVCF
|
6.3 | IC50 | 2 | — | |
MQSHODMZMFZJNV
|
6.3 | IC50 | 2 | — | |
NCWNVZMHTRKEOP
|
6.3 | IC50 | 2 | — | |
NCWNVZMHTRKEOP
|
6.3 | IC50 | 3 | — | |
NKTVKMCHRMDFHV
|
6.3 | IC50 | 5 | — | |
NVTDZAFTCNOHHZ
|
6.3 | IC50 | 2 | — | |
NXEPIACAUVNFCK
|
6.3 | IC50 | 2 | — | |
PJTDZXIEHYQSQR
|
6.3 | IC50 | 2 | — | |
QUFURWJAQILIFO
|
6.3 | IC50 | 9 | — | |
QZCWPDPWSBOTEU
|
6.3 | IC50 | 7 | — | |
REZFVUNAFUHYBW
|
6.3 | IC50 | 5 | Yes |