Target Details
| UniProt AC | P07948 |
|---|---|
| Gene Symbol | LYN |
| Protein Name | Tyrosine-protein kinase Lyn |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 474
- Clinical molecules 117
- Avg pChEMBL 6.97
KEGG Pathways (13)
- B cell receptor signaling pathway
- Chemokine signaling pathway
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- IgSF CAM signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Long-term depression
- NF-kappa B signaling pathway
- Platelet activation
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYHDXABKNJMNEZ
|
7.2 | Ki | 10 | — | |
MQRDVGBWWVWMEN
|
7.2 | Ki | 47 | — | |
NRGYZNJPCGRCLV
|
7.2 | Ki | 52 | — | |
NRZYTPAJGVTKIM
|
7.2 | Ki | 38 | — | |
NWAUBAGBGOPJLF
|
7.2 | Ki | 51 | Yes | |
NXSJMRCTGYTSTK
|
7.2 | Kd | 200 | — | |
PTVPBWWDGZSEAF
|
7.2 | Ki | 63 | — | |
UXQLMVSZSYZFID
|
7.2 | Ki | 12 | — | |
WFTZMAAMCVPJJT
|
7.2 | Ki | 26 | — | |
WZZXMNBOPNKKSX
|
7.2 | Ki | 10 | — | |
XCHWBXBDZRJVDP
|
7.2 | Ki | 51 | — | |
PTHVKCSYXICMAR
|
7.2 | IC50 | 14 | — | |
XQGUIRKPWAXDLW
|
7.2 | IC50 | 4 | — | |
SDVAHCXGDGYWFA
|
7.2 | IC50 | 12 | — | |
UKYJKXMPIDEQFF
|
7.2 | IC50 | 16 | — | |
XPIADKIXMMYTSD
|
7.2 | IC50 | 5 | Yes | |
WCSCGZHKZNEMNJ
|
7.2 | IC50 | 4 | — | |
MVYBDSJHHWQUEP
|
7.1 | IC50 | 4 | Yes | |
OPHSZSZDICRBPP
|
7.1 | IC50 | 16 | — | |
UARVSLPFGRKWQN
|
7.1 | IC50 | 11 | — | |
FCJGMZMSVIAAJU
|
7.1 | IC50 | 9 | — | |
DLPARMNJOHFOLU
|
7.1 | Ki | 14 | Yes | |
FUZSHLVNKZZEKR
|
7.1 | IC50 | 16 | — | |
LGHBDVLAHHANMX
|
7.1 | Ki | 53 | — | |
MFMXAWQGPQXDRJ
|
7.1 | Ki | 27 | — | |
MTCHQDWUHQADSY
|
7.1 | Ki | 29 | — | |
OTVCFDOYUHREFJ
|
7.1 | Ki | 26 | — | |
SFPWNTQWFFNJIH
|
7.1 | Ki | 48 | — | |
WINHZLLDWRZWRT
|
7.1 | Ki | 66 | — | |
AYZBGELVIWCHIM
|
7.1 | IC50 | 5 | Yes | |
VCIZYTQJDGPPDJ
|
7.1 | IC50 | 6 | — | |
GVRXIDPSFXZQGC
|
7.1 | IC50 | 4 | — | |
YGTYIGUWQYTZMS
|
7.1 | IC50 | 5 | Yes | |
APPXQUDJLJXULP
|
7.1 | IC50 | 47 | — | |
FNVQWFPDIYQCSF
|
7.1 | IC50 | 8 | Yes | |
PPCDZYRDXIKRDW
|
7.1 | IC50 | 6 | Yes | |
CAWABSRZIMATJO
|
7.0 | IC50 | 9 | — | |
YCGAVAFYTUFYPA
|
7.0 | IC50 | 6 | Yes | |
FLBNLJLONKAPLR
|
7.0 | Kd | 31 | — | |
AGJAPEBQOOHERM
|
7.0 | IC50 | 4 | Yes | |
BDPBZUHWAVABDM
|
7.0 | Ki | 11 | — | |
DJLORVJVWIBDME
|
7.0 | Ki | 24 | — | |
FOONBYIHFUMRSX
|
7.0 | Ki | 12 | — | |
GLDQJVYQRVZJIH
|
7.0 | IC50 | 3 | — | |
HHZIURLSWUIHRB
|
7.0 | Kd | 57 | Yes | |
HUNGUWOZPQBXGX
|
7.0 | IC50 | 4 | — | |
HXHAJRMTJXHJJZ
|
7.0 | Ki | 52 | Yes | |
JSDGKSMNPHJDFK
|
7.0 | Ki | 35 | — | |
MVJMMLFMPWITEJ
|
7.0 | Ki | 110 | — | |
MZDKLVOWGIOKTN
|
7.0 | Ki | 80 | — |