Target Details
| UniProt AC | P07948 |
|---|---|
| Gene Symbol | LYN |
| Protein Name | Tyrosine-protein kinase Lyn |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 474
- Clinical molecules 117
- Avg pChEMBL 6.97
KEGG Pathways (13)
- B cell receptor signaling pathway
- Chemokine signaling pathway
- Epithelial cell signaling in Helicobacter pylori infection
- Epstein-Barr virus infection
- Fc epsilon RI signaling pathway
- Fc gamma R-mediated phagocytosis
- IgSF CAM signaling
- Kaposi sarcoma-associated herpesvirus infection
- Lipid and atherosclerosis
- Long-term depression
- NF-kappa B signaling pathway
- Platelet activation
- Viral carcinogenesis
Associated Diseases (1)
Active Molecules (474)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZATGFXTWDKIEKC
|
7.6 | IC50 | 8 | Yes | |
YDELNSXADYPQGS
|
7.6 | IC50 | 15 | Yes | |
CRPUDAVZTZIKMJ
|
7.5 | IC50 | 7 | Yes | |
NHVGQRASKRTWLZ
|
7.5 | IC50 | 5 | Yes | |
FDVSOQRNTAPCHB
|
7.5 | IC50 | 7 | Yes | |
NJCKEVQJALLWBU
|
7.5 | IC50 | 2 | — | |
SLEWGGZPOQNVSU
|
7.5 | Kd | 22 | — | |
WVXNSAVVKYZVOE
|
7.5 | IC50 | 92 | — | |
UMBFDGUGXMOMHX
|
7.5 | IC50 | 12 | — | |
MOXXQFNQDDSJHT
|
7.5 | Ki | 6 | — | |
ZFGRQAXIHZXQBZ
|
7.5 | IC50 | 4 | Yes | |
CXBBWVXSZINRCS
|
7.5 | Ki | 41 | — | |
JBBNRIFQSNWZOK
|
7.5 | IC50 | 4 | — | |
NFKMFNBKEOQNPZ
|
7.5 | Ki | 43 | — | |
UUWNXFJBBYAMDT
|
7.5 | Ki | 46 | — | |
XKFTZKGMDDZMJI
|
7.5 | Ki | 56 | — | |
XNEPVLVYFUGJLF
|
7.5 | Ki | 27 | — | |
CXQHYVUVSFXTMY
|
7.5 | Kd | 154 | — | |
YZLKFFPFWYDBEB
|
7.5 | IC50 | 3 | — | |
ZDACFCFMMWTLTA
|
7.5 | IC50 | 9 | — | |
PGQWALGGBUYLQF
|
7.4 | IC50 | 12 | — | |
ADCQRIVAZWFZCZ
|
7.4 | IC50 | 4 | — | |
AIQDZMUPVYDVLB
|
7.4 | Ki | 48 | — | |
DKSNLQYRZJKYOC
|
7.4 | Ki | 51 | — | |
HKSZLNNOFSGOKW
|
7.4 | Kd | 213 | — | |
LRHOWQSLEKDTCW
|
7.4 | IC50 | 2 | — | |
RDNOLDWOMGZBPI
|
7.4 | IC50 | 8 | Yes | |
RKLGMDOZEOTQEM
|
7.4 | Ki | 12 | — | |
BCNXUFFSRWFFQA
|
7.4 | IC50 | 5 | Yes | |
SVYYVGZMWJYFIE
|
7.4 | IC50 | 3 | — | |
ZTMATBOBWAXBCV
|
7.4 | IC50 | 4 | — | |
YTSHBWDZKXHZDM
|
7.3 | IC50 | 2 | — | |
GWDSKGBTVQNXRT
|
7.3 | IC50 | 2 | — | |
MXJMJNRCJKHFPP
|
7.3 | IC50 | 10 | — | |
CDISOBGWDHAHGF
|
7.3 | IC50 | 16 | — | |
CNTCGRJDUJEUDG
|
7.3 | Ki | 37 | — | |
DBXOMQJZSQLQED
|
7.3 | Ki | 12 | — | |
KNACLJBHKVSTDL
|
7.3 | Ki | 40 | — | |
OEFUMBDQRIIGBZ
|
7.3 | IC50 | 3 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 15 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 13 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 6 | — | |
IBCGPVVKHZXWNX
|
7.3 | IC50 | 7 | — | |
KUCNBQPAJZRQMJ
|
7.3 | IC50 | 11 | — | |
MJQGHLODJHABRA
|
7.3 | IC50 | 10 | — | |
XYFPWWZEPKGCCK
|
7.3 | IC50 | 34 | — | |
OYAMULIHRWEUAR
|
7.2 | IC50 | 7 | Yes | |
WJEOLQLKVOPQFV
|
7.2 | Kd | 24 | — | |
DZSUJUOJJJCWGG
|
7.2 | Ki | 55 | Yes | |
HKZKELVPGXJIMW
|
7.2 | Ki | 41 | — |