Target Details
| UniProt AC | P07947 |
|---|---|
| Gene Symbol | YES1 |
| Protein Name | Tyrosine-protein kinase Yes |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 158
- Clinical molecules 54
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KTEIFNKAUNYNJU
|
6.1 | Kd | 114 | — | |
VKMLXLHRFKTEPP
|
6.1 | Ki | 2 | — | |
WVUNYSQLFKLYNI
|
6.1 | Kd | 46 | Yes | |
HXHAJRMTJXHJJZ
|
6.0 | Kd | 52 | Yes | |
YABJJWZLRMPFSI
|
6.0 | Kd | 34 | — | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.0 | Kd | 91 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — |