Target Details
| UniProt AC | P07947 |
|---|---|
| Gene Symbol | YES1 |
| Protein Name | Tyrosine-protein kinase Yes |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 158
- Clinical molecules 54
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JOOXLOJCABQBSG
|
6.9 | Kd | 139 | — | |
UHTHHESEBZOYNR
|
6.9 | Kd | 66 | Yes | |
WINHZLLDWRZWRT
|
6.9 | Kd | 201 | Yes | |
TXGKRVFSSHPBAJ
|
6.9 | IC50 | 11 | — | |
ZGBGPEDJXCYQPH
|
6.9 | IC50 | 3 | — | |
RMTJSBZCZKCYHB
|
6.8 | IC50 | 13 | — | |
DDQFACKDLYLRGU
|
6.8 | IC50 | 5 | Yes | |
MFAQYJIYDMLAIM
|
6.8 | Kd | 130 | Yes | |
MGGBYMDAPCCKCT
|
6.8 | IC50 | 23 | — | |
UIARLYUEJFELEN
|
6.8 | Kd | 289 | Yes | |
XZIADLYCTOCKRV
|
6.8 | IC50 | 5 | — | |
ALKJNCZNEOTEMP
|
6.8 | Kd | 55 | — | |
SLEWGGZPOQNVSU
|
6.8 | Kd | 22 | — | |
VTJHGMZHVOXJPG
|
6.7 | IC50 | 15 | — | |
JWNPDZNEKVCWMY
|
6.6 | Kd | 57 | Yes | |
MHXGEROHKGDZGO
|
6.6 | IC50 | 10 | — | |
JCJSAFZMXVQVBR
|
6.6 | IC50 | 11 | Yes | |
CTNPALGJUAXMMC
|
6.6 | Kd | 151 | — | |
HHFBDROWDBDFBR
|
6.6 | Kd | 40 | Yes | |
ODPGGGTTYSGTGO
|
6.6 | Kd | 153 | — | |
WDTHDWKPTWWHLS
|
6.6 | IC50 | 13 | — | |
XXJWYDDUDKYVKI
|
6.6 | Kd | 52 | — | |
KCEWOOVCWCPFCY
|
6.5 | IC50 | 5 | — | |
UWXSAYUXVSFDBQ
|
6.5 | Kd | 6 | — | |
USVCWSAJUAARAL
|
6.5 | Kd | 8 | — | |
APPXQUDJLJXULP
|
6.4 | IC50 | 47 | — | |
DZFZXPPHBWCXPQ
|
6.4 | Kd | 12 | — | |
GUBJNPWVIUFSTR
|
6.4 | Kd | 103 | — | |
WMMNTQFZCHUZSM
|
6.4 | IC50 | 14 | — | |
AKSZNKRUJCTEIJ
|
6.4 | IC50 | 4 | — | |
BLQYVHBZHAISJM
|
6.4 | Kd | 21 | Yes | |
IAYGCINLNONXHY
|
6.4 | Kd | 50 | — | |
GCIKSSRWRFVXBI
|
6.3 | Kd | 109 | Yes | |
HKKYOSCAKSXOJA
|
6.3 | IC50 | 3 | — | |
PYCBKUUFGVDPOF
|
6.3 | Ki | 4 | — | |
RERCSHBOJZUUMN
|
6.3 | IC50 | 2 | — | |
ILWOIMOKLTUADE
|
6.3 | IC50 | 4 | — | |
IKLGYJACVCXYIL
|
6.3 | IC50 | 5 | — | |
NKTVKMCHRMDFHV
|
6.3 | IC50 | 5 | — | |
RSWVUHGRSKMXFQ
|
6.3 | IC50 | 3 | — | |
PABMYTICQCKZAG
|
6.2 | IC50 | 3 | — | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes | |
WJEOLQLKVOPQFV
|
6.2 | Kd | 24 | — | |
NXSJMRCTGYTSTK
|
6.2 | Kd | 200 | — | |
PFTXFNSHFZLJNT
|
6.2 | IC50 | 17 | — | |
CDBACQLZGUZJLV
|
6.2 | IC50 | 2 | — | |
DMXWTHVOLSODIU
|
6.2 | Ki | 4 | — | |
YFNWWNRZJGMDBR
|
6.2 | Kd | 35 | — | |
UHIZYQVRKSWIFO
|
6.1 | Kd | 3 | — | |
UORAPQCBWYIISR
|
6.1 | IC50 | 15 | — |