Target Details
| UniProt AC | P07947 |
|---|---|
| Gene Symbol | YES1 |
| Protein Name | Tyrosine-protein kinase Yes |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 158
- Clinical molecules 54
- Avg pChEMBL 7.39
KEGG Pathways (1)
Active Molecules (158)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AILRADAXUVEEIR
|
7.7 | IC50 | 75 | — | |
IRBVGTPPFBYDKX
|
7.7 | IC50 | 9 | — | |
LOGJQOUIVKBFGH
|
7.7 | IC50 | 11 | Yes | |
NDEXUOWTGYUVGA
|
7.7 | IC50 | 12 | — | |
VJMLVRWRSSMUGF
|
7.7 | IC50 | 6 | Yes | |
VTMJLOMESRVYBL
|
7.7 | IC50 | 5 | Yes | |
WJAKMUHDSIHSPY
|
7.7 | IC50 | 6 | Yes | |
JUSWPUDQOKINJO
|
7.7 | IC50 | 16 | — | |
NYEBJLYZEHKODB
|
7.7 | IC50 | 5 | Yes | |
WKDACQVEJIVHMZ
|
7.7 | Kd | 46 | — | |
QQWUGDVOUVUTOY
|
7.6 | Kd | 231 | Yes | |
LOLPPWBBNUVNQZ
|
7.6 | IC50 | 97 | Yes | |
XHHRGYCOEVNAKV
|
7.6 | Ki | 6 | Yes | |
KUCNBQPAJZRQMJ
|
7.6 | IC50 | 11 | — | |
CFIIVSLTMJHIQA
|
7.5 | IC50 | 3 | Yes | |
FTDWSWREBGYXDZ
|
7.5 | IC50 | 10 | — | |
FUZSHLVNKZZEKR
|
7.5 | IC50 | 16 | — | |
UQIPWVWRJALLFY
|
7.5 | IC50 | 5 | Yes | |
YAAKXNXVUNFSPT
|
7.5 | IC50 | 5 | Yes | |
LSJWYMSFUWBGPN
|
7.5 | IC50 | 17 | — | |
CDISOBGWDHAHGF
|
7.5 | IC50 | 16 | — | |
NHHQJBCNYHBUSI
|
7.5 | Kd | 220 | — | |
ZVPDNRVYHLRXLX
|
7.4 | IC50 | 35 | Yes | |
OPHSZSZDICRBPP
|
7.4 | IC50 | 16 | — | |
GHWPJPRJEAOHFY
|
7.4 | IC50 | 6 | Yes | |
OOMBFNDWQIGHEK
|
7.4 | Kd | 22 | — | |
PUWQBZYOEYJCIO
|
7.4 | IC50 | 6 | Yes | |
XYFZVVYVIFJBIS
|
7.4 | IC50 | 17 | — | |
PGQWALGGBUYLQF
|
7.4 | IC50 | 12 | — | |
AYCPARAPKDAOEN
|
7.3 | IC50 | 73 | — | |
CXQHYVUVSFXTMY
|
7.3 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.3 | Kd | 149 | — | |
HKSZLNNOFSGOKW
|
7.3 | Kd | 213 | — | |
UORAPQCBWYIISR
|
7.3 | IC50 | 13 | — | |
OMIQRSKHABIPRH
|
7.3 | IC50 | 15 | — | |
KZRDVFBPXXGSPD
|
7.3 | IC50 | 9 | — | |
MJQGHLODJHABRA
|
7.3 | IC50 | 10 | — | |
QUFURWJAQILIFO
|
7.3 | IC50 | 9 | — | |
XKFTZKGMDDZMJI
|
7.3 | Kd | 64 | Yes | |
OSAWFUCUZJNEID
|
7.2 | IC50 | 20 | — | |
GZYUJXFTHLKPAK
|
7.2 | IC50 | 16 | — | |
QZCWPDPWSBOTEU
|
7.2 | IC50 | 7 | — | |
LAUHLGUSVSJYCI
|
7.1 | IC50 | 16 | — | |
XHBVYDAKJHETMP
|
7.1 | IC50 | 24 | Yes | |
BOWYXGHFMQMXPT
|
7.1 | Ki | 9 | — | |
XZXHXSATPCNXJR
|
7.1 | Kd | 165 | Yes | |
LXURGGKEOPHREO
|
7.1 | IC50 | 13 | — | |
FLBNLJLONKAPLR
|
7.0 | Kd | 31 | — | |
CEUSZLVORFRBCV
|
7.0 | IC50 | 13 | — | |
ZUMICAGHFTUJTI
|
7.0 | IC50 | 4 | Yes |